|
2016 |
|
 |
P Khare, S Jagtap, Y Jain, RK Baboota, P
Mangal, RK Boparai, KK Bhutani, SS Sharma, LS Premkumar, KK
Kondepudi, K Chopra, M Bishnoi. Cinnamaldehyde
supplementation prevents fasting-induced hyperphagia, lipid
accumulation, and inflammation in high-fat diet-fed mice.
Biofactors 2016, 42, 201-11. |
 |
P Mangal, P Khare, S Jagtap, M Bishnoi, KK
Kondepudi, KK Bhutani. Screening of six Ayurvedic medicinal
plants for anti-obesity potential: An investigation on
bioactive constituents from Oroxylum indicum (L.) Kurz bark.
Journal of Ethanopharmacology 2016, pii:
S0378-8741(16)30498- 6. |
 |
S Jagtap, P Khare, P Mangal, KK Kondepudi, M
Bishnoi, KK Bhutani. Effect of mahanimbine, an alkaloid from
curry leaves, on high fat diet induced adiposity, insulin
resistance and inflammatory alterations. Biofactors
2016 (Accepted). |
|
 |
Jagtap S, Khare P, Mangal P,
Kondepudi KK, Bishnoi M and Bhutani KK. Protective effects
of phyllanthin, a lignin from Phyllanthus amarus, against
induced metabolic disturbances in mice. RSC Adv.
2016, (DoI: 10.1039/C6RA10774E). |
|
 |
Kuppala R, Govindarajan M,
Tambat R, Patel N, Nandanwar H, Bhutani KK and Kartha KP.
Synthesis and antibacterial activity of ricinoleic acid
glycosides. RSC Adv. 2016, 6:3700-13. |
|
 |
Singh S. Stability Testing During Development
of Nanopharmaceuticals. Pharmaceutical Nanotechnology
2016, 3(4): 306-14. |
|
 |
Sahu A, Narayanam M, Kurmi M, Ladumor M and
Singh S. Quantitation of Memantine Hydrochloride Bulk Drug
and its Marketed Formulations Using Proton Nuclear Magnetic
Resonance Spectrometry. Magnetic Resonance in
Chemistry 2016, 54(8):632-36. |
|
 |
Kurmi M, Singh DK, Tiwari S, Sharma P and
Singh S.
Stability behaviour of antiretroviral drugs and their
combinations. 3: Characterization of interaction products of
emtricitabine and tenofovir disoproxil fumarate by mass
spectrometry. Journal
of Pharmaceutical and Biomedical Analysis
2016, 128: 438–46. |
|
 |
Kurmi M,
Kushwah BS, Sahu A,
Narayanam
M and Singh S. Stability
Behaviour of Antiretroviral Drugs and their Combinations. 2:
Characterization of Interaction Products of Lamivudine and
Tenofovir Disoproxil Fumarate by Mass and NMR Spectrometry.
Journal of Pharmaceutical and Biomedical
Analysis
2016,
125:
245–59. |
|
 |
Parmar K, Jhajra S
and Singh S. Detection of
Glutathione Conjugates of Amiodarone and Its Reactive
Diquinone Metabolites in Rat Bile Using Mass Spectrometry
Tools. Rapid Communications in Mass Spectrometry
2016,
30(10): 1242–48. |
|
 |
Singh DK, Kurmi M, Handa T and
Singh S.
LC-MS/TOF, LC-MSn and H/D Exchange Studies on
Solifenacin Succinate Targeted to Characterize its Forced
Degradation Products.
Chromatographia 2016,
79(3):
159-68. |
|
 |
Jhajra S and Singh S. Identification of
Stable and Reactive Metabolite(S) of Nelfinavir In Human
Liver Microsomes and rCYP3A4. Journal of
Pharmaceutical and Biomedical Analysis 2016, 118:
214–27. |
|
 |
Ladumor M, Tiwari S, Patil A, Bhavsar K,
Jhajra S, Prasad B and Singh S.
High-resolution mass spectrometry in
metabolite identification. In: Comprehensive
Analytical chemistry 2016: Applications of TOF and
Orbitrap MS in Environmental, Food, Doping, and Forensic
Analysis, Sandra Pérez,
Peter Eichhorn, and Damia Barcelo Culleres, (Eds.),
Elsevier. Vol. 71. |
|
 |
Bansal S, Maurya IK, Yadav N,
Thota CK, Kumar V, Tikoo K, Chauhan VS and Jain R.
C-Terminal fragment, Ab32-37 analogues protect against A?
aggregation-induced toxicity. ACS Chem. Neurosci.
2016, 7: 615-23. |
|
 |
Meena CL, Thakur A, Nandekar
PP, Sharma SS, Sangamwar AT and Jain R. Synthesis and
biology of ring-modified L-histidine containing thyrotropin-releasing
hormone (TRH) analogues.
European Journal of Medicinal Chemistry 2016, 111: 72-83. |
|
 |
Mittal S, Kaur S, Swami A,
Maurya IK, Jain R, Wangoo N and Sharma RK. Alkylated
histidine based short cationic antifungal peptides:
synthesis, biological evaluation and mechanistic
investigations. RSC Adv. 2016, 6: 41951-61. |
|
 |
Kaur S, Bhararia A, Sharma KK,
Mittal S, Jain R, Wangoo N and Sharma RK. Thyrotropin-releasing
hormone loaded and chitosan engineered polymeric
nanoparticles: towards effective delivery of neuropeptides.
J Nanosci. Nanotechnol. 2016, 16: 5324-32. |
|
 |
Nandekar PP, Khomane K, Chaudhary V, Rathod
VP, Borkar RM, Bhandi MM, Srinivas R, Sangamwar AT, Guchhait
SK and Bansal AK. Identification of Leads for
Antiproliferative Activity on MDA-MB-435 Human Breast Cancer
Cells through Pharmacophore and CYP1A1-mediated Metabolism. European
Journal of Medicinal Chemistry 2016, 115: 82-93. |
|
 |
Sheokand S, Modi SR and Bansal AK. Quantification
of low levels of amorphous content in crystalline celecoxib
using dynamic vapor sorption (DVS). European Journal
of Pharmaceutics and Biopharmaceutics 2016, 102:
77-86. |
|
 |
Shete GB and Bansal AK. NanoCrySP
Technology for Generation of Drug Nanocrystals:
Translational Aspects and Business Potential. Drug
Delivery and Translational Research
2016,
6: 392-98. |
|
 |
Sharma RJ, Gupta RC, Singh S, Bansal AK and
Singh IP. Stability of anthocyanins- and anthocyanidins-
enriched extracts, and formulations of fruit pulp of Eugenia
jambolana ('Jamun'). Food Chemistry 2016, 190:
808-17. |
|
 |
Jawale A, Datusalia AK, Bishnoi M and Sharma
SS. Reversal of Diabetes-induced Behavioral and Neurochemical Deficits by Cinnamaldehyde.
Phytomedicine 2016, 23(9): 923-30. |
|
 |
Bajaj P, Agarwal G, Tripathy R, Datusalia AK,
Sharma SS and Pande A. Refolded recombinant human
paraoxonase 1 variant exhibits prophylactic activity against
organophosphate poisoning. Applied Biochemistry and
Biotechnology 2016 (in
press). |
|
 |
Das NR and Sharma SS.
Cognitive Impairment Associated with
Parkinson’s Disease: Role of Mitochondria. Current
Neuropharmacology 2015.
DOI: 10.2174/1570159X14666160104142349)
(in press). |
|
 |
Komirishetty P, Areti A, Yerra VG, Ruby PK, Sharma SS,
Gogoi R, Sistla R and Kumar A. PARP inhibition attenuates
neuroinflammation and oxidative stress in chronic
constriction injury induced peripheral neuropathy.
Life Sciences 2016, 150: 50–60. |
|
 |
Negi G,
Vanaja N, Kamble P and Sharma SS. Heme oxygenase-1, a
novel target for the treatment of diabetic complications:
focus on diabetic peripheral neuropathy.
Pharmacological Research 2016,
102:158-167. |
|
 |
O’Donnell JN,
Gulati A, Lavhale MS, Sharma SS, Patel AJ, Rhodes NJ and
Scheetz MH.
Pharmacokinetics
of centhaquin citrate in a rat model.
Journal of Pharmacy and Pharmacology 2016, 68(1):56-62. |
|
 |
Datusalia
A, and Sharma SS. NF-κB Inhibition Resolves Cognitive
Deficits in Experimental Type 2 Diabetes Mellitus through
CREB and Glutamate/GABA Neurotransmitters Pathway.
Current Neurovascular Research 2016, 13(1):22-32. |
|
 |
Chaudhary V, Venghateri
JB, Dhaked
HPS, Bhoyar
AS, Guchhait
SK and Panda D.
Novel Combretastatin-2-aminoimidazole
Analogues as Potent Tubulin Assembly Inhibitors: Exploration
of Unique Pharmacophoric Impact of Bridging Skeleton and
Aryl Moiety.
Journal of Medicinal Chemistry
2016, 59: 3439-51. |
|
 |
Guchhait
SK, Chaudhary V, Rana
VA, Priyadarshani G, Kandekar S and Kashyap
M. Oxidative Dearomatization of Indoles via
Pd-Catalyzed C−H Oxygenation: An Entry to C2-Quaternary
Indolin-3-ones.
Organic Letters
2016, 15: 1534-37. |
|
 |
Priyadarshani G, Amrutkar S, Nayak A,
Banerjee UC,
Kundu CN, Guchhait
SK. Scaffold-hopping of bioactive flavonoids:
Discovery of aryl-pyridopyrimidinones as potent anticancer
agents that inhibit catalytic role of
topoisomerase IIa.
European Journal of Medicinal Chemistry
2016, 122: 43-54. |
|
 |
Guchhait
SK, Priyadarshani G and
Gulghane NM.
A reaction of 1,2-diamines and aldehydes with
silyl cyanide as cyanide pronucleophile to access
2-aminopyrazines and 2-aminoquinoxalines.
RSC Advances
2106, 6: 56056-63. |
|
 |
Gani Z, Boradia VM, Ram
JR, Suryavanshi PM, Patil P, Kumar S , Singh R, Raje M and
Raje CI. Purification and Characterization of
Glyceraldehyde-3-phosphate-dehydrogenase (GAPDH) from Pea
Seeds.
Prt. Exp
Pur. 2016, DOI: 10.1016/j.pep.2016.06.014. |
|
 |
Sheokand N, Malhotra H,
Chauhan AS, Kumar M, Chaudhary S, Patidar A, Boradia VM,
Raje CI and Raje M. Reverse overshot water-wheel
retroendocytosis of Apo Transferrin extrudes cellular iron.
J Cell Sci. 2016, 129(4): 843-53. DOI: 10.1242/jcs.180356. |
|
 |
Kaur PK, Tripathi N, Desale J, Neelagiri S,
Yadav S, Bharatam PV and Singh S. Mutational and Structural
Analysis of Conserved Residues in Ribose-5-Phosphate
Isomerase B from Leishmania donovani: Role in Substrate
Recognition and Conformational Stability.
PLoS ONE
2016, 11(3): e0150764. |
|
 |
Soumya N, Tandan H, Damre MV, Gangwal RP,
Sangamwar AT and Singh S. Leucine-684: A conserved residue
of an AMP-acetyl CoA synthetase (AceCS) from Leishmania
donovani is involved in substrate recognition, catalysis and
acetylation.
Gene
2016, 580(2): 125-33. |
|
 |
Lunagariya NA, Gohil VM, Kushwah V, Neelagiri
S, Jain S, Singh S and Bhutani KK. Design, synthesis and
biological evaluation of 1,3,6-trisubstituted
â-carboline
derivatives for cytotoxic and anti-leishmanial potential.
Bioorg Med Chem Lett.
2016, 26(3): 789-94. |
|
 |
Aggarwal G, Prajapati R, Tripathy RK,
Bajaj P, Iyengar ARS, Sangamwar AT and Pande AH. Toward
understanding the catalytic mechanism of human paraoxonase
1: Site specific mutagenesis at position 192.
PLoS ONE
2016, 11(2): e0147999. DOI:
10.1371/journal.pone.0147999 |
|
 |
Tripathi SP, Prajapati R, Verma N and
Sangamwar AT. Predicting substrate selectivity between
UGT1A9 and UGT1A10 using molecular modelling and molecular
dynamics approach. J Molecular Simulation
2016, 42(4): 270-288. |
|
 |
Kesharwani SS, Nandekar
PP, Pragyan
P, Rathod
V, Sangamwar
AT. Characterization of
differences in substrate specificity among CYP1A1, CYP1A2
and CYP1B1: an integrated approach employing molecular
docking and molecular dynamics simulations. J. Mol. Recognit. 2016, Feb 25.
DOI: 10.1002/jmr.2537. |
|
 |
Rathod
V, Belekar V, Garg P and Sangamwar AT. Classification of human
pregnane X receptor (hPXR) activators and non activators by
machine learning techniques: A multifaceted approach.
Comb. Chem High Throughput Screen 2016, Mar 16. |
 |
Jena SK and Sangamwar AT. Polymeric micelles
of amphiphilic graft copolymer of alpha tocopherol
succinate-g-carboxymethyl chitosan for tamoxifen delivery:
Synthesis, characterization and in vivo pharmacokinetic
study. Carbohydrate Polymers 2016, DOI:
10.1016/j.carbpol.2016.06.078. |
|
 |
Bansal D, Gudala K, Azad C and Anil D.
Predictors of Health Related
Quality of Life in Childhood Epilepsy and Comparison with
Healthy Children: Findings from Indian Study.
Turk J
Med Sci. 2016 (in-press). |
|
 |
Mullapudi A, Gudala K, Boya CS and
Bansal D. Risk of Parkinson’s Disease in the Users of
Antihypertensive Agents: An Evidence from the Meta-Analysis
of Observational Studies. J Neurodegener Dis.
2016, 2016:1-8. |
|
 |
Gudala K, Ghai B and Bansal D. Challenges in
using Symptoms Based Screening Tools while Assessing
Neuropathic Pain Component in Patients with Chronic Low Back
Pain. J Clin. Diagn. Res. 2016, 10:UL02-UL03. |
|
 |
Bansal D, Gudala K, Lavudiya S, Ghai B and
Arora P. Translation, Adaptation, and Validation of Hindi
Version of the Pain Catastrophizing Scale in Patients with
Chronic Low Back Pain for Use in India. Pain Medicine
2016, 2016:103. |
 |
Kondal A, Krishna GVM and Bansal D. Clinical
Trial Regulations in India: Progress and Challenges Arising
from Recent Amendments to Schedule Y of the Drugs and
Cosmetics (D&C) Act 1940 (D&C Rules 1945).
Pharmaceutical Medicine 2016,
30:1-13. |
 |
Golla VM, Kurmi M, Shaik K, Singh S.
Stability Behaviour of Antiretroviral Drugs and their
Combinations. 4: Characterization of Degradation Products of
Tenofovir Alafenamide Fumarate and Comparison of its
Degradation and Stability Behaviour with Tenofovir
Disoproxil Fumarate. Journal
of Pharmaceutical and Biomedical Analysis
2016,
131:146–55. |
 |
Sahu A,
Narayanam M, Kurmi M, Ladumor M, Singh S. Quantitation of
Memantine Hydrochloride Bulk Drug and its Marketed
Formulations Using Proton Nuclear Magnetic Resonance
Spectrometry. Magnetic Resonance in Chemistry
2016, 54(8): 632-6. |
 |
Kurmi M, Singh DK, Tiwari S, Sharma P, Singh
S. Stability
behaviour of antiretroviral drugs and their combinations. 3:
Characterization of interaction products of emtricitabine
and tenofovir disoproxil fumarate by mass spectrometry,
Journal of
Pharmaceutical and Biomedical Analysis
2016, 128: 438–46. |
 |
Kurmi M,
Kushwah BS, Sahu A,
Narayanam
M and Singh S. Stability
Behaviour of Antiretroviral Drugs and their Combinations. 2:
Characterization of Interaction Products of Lamivudine and
Tenofovir Disoproxil Fumarate by Mass and NMR Spectrometry.
Journal of Pharmaceutical and Biomedical
Analysis
2016, 125:
245–59. |
 |
Parmar K, Jhajra S,
Singh S. Detection of
Glutathione Conjugates of Amiodarone and Its Reactive
Diquinone Metabolites in Rat Bile Using Mass Spectrometry
Tools, Rapid Communications in Mass Spectrometry
2016, 30(10): 1242–8. |
 |
Singh DK, Kurmi M, Handa T,
Singh S.
LC-MS/TOF, LC-MSn and H/D Exchange Studies on
Solifenacin Succinate Targeted to Characterize its Forced
Degradation Products,
Chromatographia 2016,
79(3):159-68. |
 |
Jhajra S and Singh S. Identification of
Stable and Reactive Metabolite(S) of Nelfinavir In Human
Liver Microsomes and rCYP3A4,
Journal of Pharmaceutical and Biomedical Analysis
2016,
118:
214–27. |
 |
Ladumor M, Tiwari S, Patil A, Bhavsar K,
Jhajra S, Prasad B and Singh S.
High-resolution mass spectrometry in
metabolite identification, In: Comprehensive
Analytical chemistry, Vol. 71: Applications of TOF
and Orbitrap MS in Environmental, Food, Doping, and Forensic
Analysis, Sandra Pérez,
Peter Eichhorn, and Damia Barcelo Culleres, (Eds.),
Elsevier, 2016. |
 |
Singh S. Stability Testing During Development
of Nanopharmaceuticals. Pharmaceutical Nanotechnology
2016, 3(4): 306-14. |
 |
Singh S. Skill Development and
Pharmaceutical Education. APTI Bulletin 2016,
17(102): 8-17. |
 |
Thakur NS, Dwivedee BP, Banerjee UC and
Bhaumik J .Bioinspired Synthesis of Silver Nanoparticles:
Characterization, Mechanism And Applications, “Silver
Nanoparticles for Antibacterial Devices: Biocompatibility
and Toxicity", CRC Press (Tailor and Francis),
ISBN:9781498725323 (In Press) |
 |
Kumar R, Banoth L,
Banerjee UC
Kaur J Enantiomeric separation of
pharmaceutically important drug intermediates using a
Metagenomic lipase and optimization of its large scale
production. International Journal of Biological
Macromolecules 2017, 95: 995-1003. |
 |
Patel G, Patil MD, Soni S, Chisti Y and
Banerjee UC. Production of mycophenolic acid by
Penicillium brevicompactum using solid state
fermentation. Applied Biochemistry and Biotechnology
(in press) 2016. |
 |
Patel G, Patil MD, Soni S, Chisti Y and
Banerjee UC. Production of mycophenolic acid by
Penicillium brevicompactum using solid state
fermentation. Applied Biochemistry and Biotechnology
(in press) 2016. |
 |
Mulik S, Ghosh S, Bhaumik J and Banerjee UC.
Biocatalytic synthesis of (S)-Practolol, a selective
β-blocker. Biocatalysis 2016, 1(1): 130-40. |
 |
Bhaumik J, Gogia G, Kirar S, Vijay L, Thakur
NS, Banerjee UC and Laha JK. Bioinspired
Nanophotosensitizers: Synthesis and Characterization of
Noble Metal Nanoparticle-Porphyrin Conjugates. New
Journal of Chemistry 2016, 40: 724-31. |
 |
Ghosh S, Bhaumik J, Banoth L and Banerjee
UC. Chemoenzymatic Route for the Synthesis of (S)-Moprolol,
a Potential β-Blocker, Chirality 2016, 28:
313-318 |
 |
Darpan, Joshi G, Amrutkar SM, Baviskar AT,
Kler H, Singh S, Banerjee UC, Kumar R. Synthesis and
biological evaluation of new 2, 5-dimethylthiophene/furan
based N-acetyl pyrazolines as selective topoisomerase II
inhibitors. RSC
Advances
2016, 6: 14880-92. |
 |
Mittal A, Thanki K, Jain S, Banerjee UC.
Comparative studies of anticancer and antimicrobial
potential of bioinspired silver and silver-selenium
nanoparticles. Applied Nanomedicine 2016,
1:1-6. |
 |
Patil MD, Bhaumik J, Babykutty S, Banerjee UC
and Fukumura D, Arginine Dependence of Tumor Cells:
Targeting a Chink in Cancer’s Armor. Nature Oncogene
2016, 35: 4957-72. |
 |
Patil MD, Shinde KD, Patel G, Chisti Y and
Banerjee UC. Use of response surface method for
maximizing the production of arginine deiminase by
Pseudomonas putida. Biotechnology Reports
2016, 10: 29-37. |
 |
Thakur NS, Bhaumik J, Sooram B, Banoth L and
Banerjee UC.
Synthesis of enantiopure drugs and drug
intermediates using In silico generated archetype
biocatalyst-A case study using Alprenolol as a model drug.
ChemistrySelect
2016 1: 871-76. |
 |
Ajayi EIO, Modo EU, Adebamowo AO,
Banerjee UC, Tewe OO and Olorunsogo OO,
Inhibitory activity of ethanol extract of Manihot
esculenta on mitochondrial membrane permeability
transition pore and caspase 3 in Type 2 diabetes mellitus.
International Journal of Biochemistry Research &
Review 2016, 9(4): 1-10. |
 |
Sawant G, Ghosh S, Banesh S,
Bhaumik J
and Banerjee UC.
In-silico approach
towards lipase mediated chemoenzymatic synthesis of (S)-Ranolazine,
as an anti-anginal drug. RSC
Advances
2016, 6: 49150-7. |
 |
Ghosh S, Mohan U,
Banerjee UC.
Studies on the production of shikimic acid using the aroK
knockout strain of Bacillus megaterium. World
Journal of Microbiology and Biotechnology 2016, 32:
1-11. |
 |
Priyadarshani G, Amrutkar S, Nayak A,
Banerjee UC,
Kundu CN, Guchhait SK Scaffold-hopping of bioactive
flavonoids: Discovery of aryl-pyridopyrimidinones as potent
anticancer agents that inhibit catalytic role of
topoisomerase IIα, European Journal of Medicinal
Chemistry 2016,
122: 43-54. |
 |
Priyadarshani G,
Nayak A, Amrutkar SM, Das S, Guchhait SK, Kundu
CK and Banerjee UC.
Scaffold-Hopping of Natural Bioactive Aurones:
Identification of 2-Arylideneimidazo[1,2-a]pyridinones
as Potent Topoisomerase IIα-inhibiting Anticancer Agents.
ACS Medicinal Chemistry Letters
2016, 7: 1056–61. |
 |
Patel G, Patil MD, Soni S, Khobragade TP,
Chisti Y and Banerjee UC. Production of mycophenolic acid
by Penicillium brevicompactum – a comparison of two
methods of optimization.
Biotechnology Reports
2016, 11: 77-85. |
 |
Chauhan M, Joshi G, Kashyap A, Amrutkar SM,
Banerjee UC,
Singh S, Bhilare K, Kumar R Dual inhibitors of epidermal
growth factor receptor and topoisomerase IIα derived from
quinoline scaffold. RSC Advances 2016, 6:
77717-34. |
 |
Ghoshal G, Shivhare US and
Banerjee UC.
Thermo-mechanical and Micro-structural
Properties of Xylanase Containing Whole Wheat Bread,
Food Science and Human Wellness 2016, 5: 219-29. |
 |
Patil MD, Patel G, Surywanshi B, Shaikh N,
Garg P, Chisti Y, Banerjee UC. Disruption of Pseudomonas
putida by high pressure homogenization: a comparison of
the predictive capacity of three process models for the
efficient release of arginine deiminase. AMB Express
2016, 6: 84. |
 |
Sharma KK, Mandloi M, Rai N,
Jain R. Copper-catalyzed N-(hetero)arylation of amino acids
in water. RSC Adv. 2016, 6, 96762-67. |
 |
Mittal S, Maurya IK, Kaur S,
Swami A, Jain, R, Wangoo N, Sharma RK. Insights into
mechanistic and synergistic aspects of novel synthetic short
cationic antibacterial peptides. ChemistrySelect
2016, 1:5510-16. |
 |
Rajput SK, Sharma AK, Meena
CL, Pant AB, Jain R, Sharma SS. Effect of L-pGlu-(1-benzyl)-L-His-L-Pro-NH2
against in-vitro and in-vivo models of cerebral ischemia and
associated neurological disorders. Biomed.
Pharmacother. 2016, 84:1256-65. |
 |
Sharma KK, Mandloi M, Jain R.
Regioselective copper-catalyzed N(1)-(hetero)arylation of
protected histidine. Org. Biomol. Chem.
2016, 14: 8937-41. |
 |
Bansal S, Maurya IK, Yadav N,
Thota CK, Kumar V, Tikoo K, Chauhan VS, Jain R. C-Terminal
fragment, A?32-37 analogues protect against A?
aggregation-induced toxicity. ACS Chem. Neurosci.
2016, 7: 615-23. |
 |
Meena CL, Thakur A, Nandekar
PP, Sharma SS, Sangamwar AT, Jain R. Synthesis and biology
of ring-modified L-histidine containing thyrotropin-releasing
hormone (TRH) analogues. Eur. J. Med. Chem.
2016, 111:72-83. |
 |
Mittal S, Kaur S, Swami A,
Maurya IK, Jain R, Wangoo N, Sharma RK. Alkylated histidine
based short cationic antifungal peptides: synthesis,
biological evaluation and mechanistic investigations.
RSC Adv. 2016, 6: 41951-61. |
 |
Kaur S, Bhararia A, Sharma KK,
Mittal S, Jain R, Wangoo N, Sharma RK. Thyrotropin-releasing
hormone loaded and chitosan engineered polymeric
nanoparticles: towards effective delivery of neuropeptides.
J. Nanosci. Nanotechnol. 2016, 16: 5324-32. |
 |
Nandekar PP, Khomane K, Chaudhary V, Rathod
VP, Borkar RM, Bhandi MM, Srinivas R, Sangamwar AT, Guchhait
SK and Bansal AK. Identification of Leads for
Antiproliferative Activity on MDA-MB-435 Human Breast Cancer
Cells through Pharmacophore and CYP1A1-mediated Metabolism. European
Journal of Medicinal Chemistry 2016, 115: 82-93. |
 |
Sheokand S, Modi SR and Bansal AK. Quantification
of low levels of amorphous content in crystalline celecoxib
using dynamic vapor sorption (DVS). European Journal
of Pharmaceutics and Biopharmaceutics 2016, 102:
77-86. |
 |
Shete GB and Bansal AK. NanoCrySP
Technology for Generation of Drug Nanocrystals:
Translational Aspects and Business Potential. Drug
Delivery and Translational Research
2016, 6: 392-8. |
 |
Sharma RJ, Gupta RC, Singh S, Bansal AK,
Singh IP. Stability of anthocyanins- and anthocyanidins-
enriched extracts, and formulations of fruit pulp of Eugenia
jambolana ('Jamun'). Food Chemistry 2016, 190:
808-17. |
 |
Khurana RK, Bansal A, Beg S, Burrow AJ,
Katare OP, Singh KK, and Singh B. Enhancing
biopharmaceutical attributes of phospholipid complex-loaded
nanostructured lipidic carriers of mangiferin: Systematic
development, characterization and evaluation.
International Journal of Pharmaceutics
2016, DOI 10.1016/j.ijpharm.2016.12.044. |
 |
Kale DP, Zode SS and Bansal AK. Challenges in
Translational Development of Pharmaceutical Cocrystals.
Journal of Pharmaceutical
Sciences 2016, DOI 10.1016/j.xphs.2016.10.021. |
 |
Thakkar S, Sharma K, Khurana S, Bansal AK.
Excipients and their Functionality for Enabling Technologies
in Oral Dosage Forms. Pharmaceutical Excipients,
Ed.: John Wiley & Sons, Inc. 2016; 97-143 |
 |
Choudhary A, Sharma RJ, Singh IP.
Quantitative analysis of major sesquiterpene lactones in
essential oil of Inula racemosa and Sausurrea
lappa using qNMR. Journal of Essential Oil Bearing
Plants 2016, 19:20-31. |
 |
Kumar R, Sethil R, Shah P, Roy I, Singh IP,
Bharatam PV, Tewari R, Garg P. Biological evaluation of
small molecule inhibitors of Mtb-ASADH enzyme. Letters
in Drug Design and Discovery 2016, 13(7):587-90. |
 |
Khan A, Bharti P, Saraf I, Mittal N, Tewari
R, Singh IP. Two new aromatic glycosides from a soil
bacterium Burkholderia gladioli OR1. Natural
Product Communications 2016, 11:663-65. |
 |
Aqil F, Jeyabalan J, Kausar H, Munagala R,
Singh IP, Gupta RC. Lung cancer inhibitory activity of
dietary berries and berry phenolics. Journal of Berry
Research 2016, 6(2):105-14. |
 |
Aqil F, Jeyabalan J, Munagala R, Singh IP,
Gupta RC. Prevention of hormonal breast cancer by dietary
jamun. Molecular Nutrition and Food Research
2016, 60(6):1470-81. |
 |
Singh V, Kahol A, Singh IP, Saraf I, Shri R.
Evaluation of antiamnesic effect of extracts of selected
Ocimum species using in vitro and in vivo
models. Journal of Ethnopharmacology 2016,
193:490-9. |
 |
Gupta S, Kumar S, Saraf I, Dhaage AH,
Upadhyay R, Chatterjee A, Singh IP. Quantification of
acetoside in Clerodendrum colebrookianum Walp. by
qNMR, HPLC and HPTLC. Trends in Carbohydrate Research
2016, 8(4):15-23. |
 |
Chaudhary V, Venghateri JB, Dhaked HPS,
Bhoyar AS, Guchhait SK and Panda D. Novel
Combretastatin-2-aminoimidazole Analogues as Potent Tubulin
Assembly Inhibitors: Exploration of Unique Pharmacophoric
Impact of Bridging Skeleton and Aryl Moiety, Journal
of Medicinal Chemistry 2016, 59: 3439-51. |
 |
Guchhait SK, Chaudhary V, Rana VA,
Priyadarshani G, Kandekar S and Kashyap M. Oxidative
Dearomatization of Indoles via Pd-Catalyzed C−H Oxygenation:
An Entry to C2-Quaternary Indolin-3-ones, Organic
Letters 2016, 15: 1534-37. |
 |
Guchhait SK, Priyadarshani G and Gulghane NM.
A reaction of 1,2-diamines and aldehydes with silyl cyanide
as cyanide pronucleophile to access 2-aminopyrazines and
2-aminoquinoxalines, RSC Advances 2016, 6:
56056-63. |
 |
Kaur PK, Tripathi N, Desale J,
Neelagiri S, Yadav S, Bharatam PV, Singh S. Mutational and
Structural Analysis of Conserved Residues in
Ribose-5-Phosphate Isomerase B from Leishmania donovani:
Role in Substrate Recognition and Conformational Stability.
PLoS One 2016, 11(3):e0150764. |
 |
Soumya N, Tandan H, Damre MV,
Gangwal RP, Sangamwar AT, Singh S. Leucine-684: A conserved
residue of an AMP-acetyl CoA synthetase (AceCS) from
Leishmania donovani is involved in substrate recognition,
catalysis and acetylation. Gene
2016,580(2):125-33. (doi: 10.1016/j.gene.2016.01.011) |
|
 |
Aggarwal
G,
Prajapati
R,
Tripathy
RK,
Bajaj
P,
Iyengar
ARS,
Sangamwar
AT,
Pande
AH.
Toward understanding the catalytic mechanism of human
paraoxonase 1: Site specific mutagenesis at position 192.
PLoS ONE
2016,
11(2): e0147999 |
|
 |
Tripathi SP, Prajapati R, Verma N and
Sangamwar AT. Predicting substrate selectivity between
UGT1A9 and UGT1A10 using molecular modelling and molecular
dynamics approach. J Molecular Simulation 2016,
42(4): 270-288J |
|
 |
Kesharwani
SS
, Nandekar
PP, Pragyan
P, Rathod
V,
Sangamwar
AT.
Characterization of differences in substrate
specificity among CYP1A1, CYP1A2 and CYP1B1: an integrated
approach employing molecular docking and molecular dynamics
simulations J Mol Recognit 2016, Feb 25. |
|
 |
Rathod
V,
Belekar
V, Garg
P and Sangamwar
AT.
Classification of human pregnane X receptor (hPXR)
activators and non activators by machine learning
techniques: A multifaceted approach.
Comb Chem High Throughput Screen. 2016,
Mar 16. |
|
 |
Jena
SK
and Sangamwar
AT.
Polymeric micelles of amphiphilic graft copolymer of alpha
tocopherol succinate-g-carboxymethyl chitosan for tamoxifen
delivery: Synthesis, characterization and in vivo
pharmacokinetic study. Carbohydrate Polymers 2016,151:1-13. |
|
 |
Daundiyal
A,
Jena
SK, Samal
SK,
Sonvane
B, Chand
M, Sangamwar
AT. Alpha lipoic acid sterylamine conjugate
based solid lipid nanoparticles for tamoxifen delivery:
Formulation, optimization, in vivo pharmacokinetic and
hepatotoxicity study J Pharm Pharmacol 2016,
68(12):1535-50. |
 |
Boradia
VM,
Patil
P,
Agnihotri
A,
Kumar
A,
Malhotra
H,
Sheokand
N,
Kumar
M,
Rajwadi
KKK,
Sahu
A,
Hasan
N,
Patkar
R,
Bhagath N, Raje
M and
Raje
CI.
Mycobacterium tuberculosis
H37Ra - a surrogate for the expression of conserved,
multimeric proteins of M.tb H37Rv. Microbial
Cell Factories. 2016 Aug 11;15(1):140.
DOI:10.1186/s12934-016-0537-0 |
 |
Gani
Z,
Boradia
VM,
Ram
JR,
Suryavanshi
PM,
Patil
P,
Kumar
S,
Singh
R,
Raje
M
and Raje
CI.
Purification and Characterization of
Glyceraldehyde-3-phosphate dehydrogenase (GAPDH) from Pea
Seeds. Protein Expression and Purification
2016, 127, 22-27, DOI 10.1016/j.pep.2016.06.014 |
 |
Sheokand
N,
Malhotra
H,
Chauhan
AS,
Kumar
M,
Chaudhary
S,
Patidar
A,
Boradia
VM,
Raje
CI,
Raje
M.
Reverse overshot water-wheel retroendocytosis of Apo
Transferrin extrudes cellular iron. Journal of Cell
Science 2016,
Feb 15;129 (4):843-853.
DOI:
10.1242/jcs.180356. |
|
2015 |
|
|
 |
Bhandari P, Kumar N, Khan MS and
Bhutani KK. Online Antioxidant
Activity and Ultra-performance
LC-Electrospray Ionization-Quadrupole
Time-of-flight Mass Spectrometry
for Chemical Fingerprinting of
Indian Polyherbal Formulations,
Natural Product Research
2015,
doi.10.1080/14786419.2015.1025231. |
|
 |
Patel NK, Khan MS, Bhutani KK.
Investigations on Leucas
Cephalotes (Roth) Spreng. For
inhibition of LPS-Induced
Pro-Inflammatory mediators in
murine macrophages and in Rat
Model. EXCLI Journal
2015, 14: 1-9. |
|
 |
Patel NK, Khan MS, Bhutani KK.
Anti-inflammatory effects of
Leucas cephalotes (Roth.) Spreng
is mediated through the
inhibition of pro-inflammatory
mediators in murine macrophages
and in rat model. EXCLI
Journal 2015, 14:
508-16. |
|
 |
Patel NK, Bairwa K, Gangwal R,
Jaiswal G, Jachak SM, Sangamwar
AT, Bhutani KK. 2'-hydroxy
flavanone derivatives as
inhibitors of pro-inflammatory
mediators: Experimental and
molecular docking studies.
Bioorganic and Medicinal
Chemistry Letters 2015,
25: 1952-5. |
|
 |
Patel NK, Jaiswal G, Bhutani KK.
A review on biological sources,
chemistry and pharmacological
activities of pinostrobin.
Natural Product Research
2015, 13:1-11. |
|
 |
Patel NK, Galipalli S, Bhutani
KK. Activity-guided
investigation on Carissa
carandas (L.) roots for
anti-inflammatory consituents.
Natural Product Research
2015, 29: 1670-2. |
|
 |
Natsume Y, Patel NNK, Tripathi
SM, Nose M, Kyuma T, Bhutani KK.
Kalyanka Ghrita: an example of
intertextuality among The Bower
Manuscript, Charak samhita,
Sushruta samhita, Astangahrdayam
samhita and Ayurvedic Formulary
of India (AFI). Indian
Journal of Traditional Knowledge
2015, 14(4): 519-24. |
|
 |
Grover J, Bhatt N, Kumar V,
Patel NK, Bondaliya BJ, Sobhia
ME, Bhutani KK, Jachak SM.
2,5-Diary1-1,3,4-oxadiazoles as
selective COX-2 inhibitors and
anti-inflammatory agents.
RSC Advances 2015, 5:
45535-44. |
|
 |
Natsume Y, Bhutani KK.
Philological study on the
history of Indian Pharmacy.
Pharmaceutical Historian
2015, 45(3): 57-63. |
|
 |
Lunagariya NA, Gohil VM, Kushwah
V, Neelagiri S, Jain S, Singh S,
Bhutani KK. Design, synthesis
and biological evaluation of
1,3,6-
trisubstituted β-carboline
derivatives for cytotoxic and
anti-leishmanial potential.
Bioorganic & Medicinal
Chemistry Letters, DOI:
10.1016/j.bmcl.2015.12.095. |
|
 |
Khare P, Jagtap S, Jain Y,
Baboota RK, Mangal P, Boparai
RN, Bhutani KK, Sharma SS,
Premkumar LS, Kondepudi KK,
Chopra K, Bishnoi M.
Cinnamaldehyde supplementation
prevents fasting-induced
hyperphagia, lipid accumulation,
and inflammation in high-fat
diet-fed miceCinnamaldehyde
supplementation prevents
fasting-induced hyperphagia,
lipid accumulation, and
inflammation in high-fat
diet-fed mice. BioFactors
2015, DOI 10.1002/biof.1265. |
|
 |
Shah PK, Kurmi M, Kumar S, Singh
S. Forced Degradation of
Lafutidine and Characterization
of its Non-Volatile and Volatile
Degradation Products Using
LC-MS/TOF, LC-MSn and
HS-GC-MS, New Journal of
Chemistry (RSC) 2015,
39:
9679–92. |
|
 |
Kurmi M, Golla VM, Kumar S, Sahu
A and Singh S. Stability
Behaviour of Antiretroviral
Drugs Alone and in Their
Combinations. 1: Characterization
of Tenofovir Disoproxil Fumarate
Degradation Products by Mass
Spectrometry,
RSC Advances
2015, 5: 96117-29. |
|
 |
Raju SPK, Narayanam M, Kumar BK,
Tejaswee S and Singh S.
Validated Stability-Indicating
Method for Alendronate Sodium
Employing Zwitterionic
Hydrophilic Interaction
Chromatography Coupled With
Charged Aerosol Detection.
Chromatographia
2015,
78 (19):1245-50. |
|
 |
Singh DK, Sahu A, Handa T,
Narayanam M, Singh S.
Comprehensive Study on Forced
Degradation Behaviour of
Prasugrel Hydrochloride by Use
of LC-MS and LC-NMR, and
Prediction of Toxicity of the
Characterized Degradation
Products. Journal of
Separation Science 2015,
38 (17):2995-3005. |
|
 |
Narayanam M, Sahu A,
Singh S. Use of
LC-MS/TOF, LC-MSn,
NMR and LC-NMR in
characterization of stress
degradation products:
Application to cilazapril.
Journal of Pharmaceutical and
Biomedical Analysis
2015, 111:190-203. |
|
 |
Jindal K, Narayanam M, Singh S.
A Systematic Strategy for the
Identification and Determination
of Pharmaceuticals in
Environment using Advanced LC–MS
Tools: Application to Ground
Water Samples. Journal of
Pharmaceutical and Biomedical
Analysis 2015, 108:
86-96. |
|
 |
Singh S.
Some
Suggestions on Conduct of
Sellable Drug Delivery Research
in Academia.
Journal of Pharmaceutical
Sciences and Technology
Management
(NMIMS, Mumbai) 2015,
1 (2): 1-7. |
|
 |
Singh S. Quality by
Design in Education (QbDE) – A
Possible Futuristic Approach to
Improve Current Status of
Pharmaceutical Education in
India. Indian Journal of
Pharmaceutical Education and
Research 2015,
49(4)(Suppl. 2): 39-45. |
|
 |
Singh S. Quality by
Design in Education (QbDE) – A
Possible Futuristic Approach to
Improve Current Status of
Pharmaceutical Education in
India. APTI Bulletin
2015, 16(95): 3-7. |
|
 |
Singh S. Including and
Emphasizing Precautions in SOPs
and STPs: An Often
Missed/Neglected Opportunity to
Communicate About Risks to Shop
Floor and Laboratory Staff in
the Pharmaceutical Industry.
Pharma Review 2015,
13(73): 63-65. |
|
 |
Tanwar B, Kumar
D, Kumar A, Ansari MI, Qadri
MM, Vaja MD, Singh M,
and Chakraborti AK.
Friedländer
annulation: Scope and
limitations of metal salt Lewis
acid catalysts in selectivity
control for the synthesis of
functionalised quinolines.
New J. Chem. 2015,
39: 9824-983. |
|
 |
Chourasiya SS,
Kathuria D, Singh S, Sonwane VC,
Chakraborti AK and Bharatam PV.
Design, Synthesis and Biological
Evaluation of Novel
Unsymmetrical Azines as Quorum
Sensing Inhibitors.
RSC
Advances
2015, DOI: 10.1039/c0xx00000x. |
|
 |
Kumar D,
Jadhavar
PS, Nautiyal M, Sharma H, Meena
PK, Adane L, Pancholia S, and
Chakraborti AK. Convenient
synthesis of 2,3-disubstituted
quinazolin-4(H)-ones and
2-styryl-3-substituted
quinazolin-4(3H)-ones:
Applications towards the
synthesis of drugs. RSC
Advances 2015, 5:
30819-825. |
|
 |
Tanwar B, Purohit
P, Raju BN, Kumar D, Kommi DN
and Chakraborti AK. An
“all-water” strategy for
regiocontrolled synthesis of
2-aryl quinoxalines. RSC
Advances 2015, 5:
11873-83. |
|
 |
Seth K, Nautiyal
M, Purohit P, Parikh N, and
Chakraborti AK. Palladium
Catalyzed Csp2-H
Activation for Direct Aryl
Hydroxylation: Unprecedented
Role of 1,4-Dioxane as Source of
Hydroxyl Radical. J. Chem.
Soc. Chem. Commun. 2015,
51: 191-4. |
|
 |
Kumar D, Kumar A,
Qadri MM, Ansari MI, Gautam A
and Chakraborti AK.
In(OTf)3-catalyzed synthesis of
2-styryl quinolines: scope and
limitations of metal Lewis acids
for tandem Friedländer
annulation–Knoevenagel
condensation. RSC Advances
2015, 5: 2920-7. |
|
 |
Singh S, Wanjari
PJ, Bhatia S, Sonwane VC,
Chakraborti AK and Bharatam PV.
Design, synthesis, biological
evaluation and toxicity studies
of N,N-disubstituted
biguanides as quorum sensing
inhibitors. Med. Chem. Res.
2015, 24: 1974-87. |
|
 |
Giri SK and
Kartha KPR. Acyl transfer
reactions of carbohydrates,
alcohols, phenols, thiols and
thiophenols under green reaction
conditions. RSC
Advances 2015,
5: 11687-96. |
|
 |
Giri SK, Narender
Y and Kartha KPR. Acyl transfer
reactions on carbohydrates:
Peracetylation, an overview. Trends
in Carbohydrate Research 2015,
7: 6-27. |
|
 |
Tyagi M, Taxak N,
Bharatam PV, Nandanwar H and
Kartha KPR. Mechanochemical
click reaction as a tool for
making carbohydrate-based
triazole-linked self-assembling
materials (CTSAMs). Carbohydrate
Research 2015,
407: 137-47. |
|
 |
Tyagi M and
Kartha KPR. Synthesis of
glycotriazololipids and
observations on their
self-assembly properties. Carbohydrate
Research2015,
413: 85-92. |
|
 |
Kuppala R,
Borrelli S, Slowski K, Sanders
DAR, Kartha
KPR and Pinto BM. Synthesis and
biological evaluation of
non-ionic substrate mimics of
UDP-Galp as
candidate inhibitors of UDP
galactopyranose mutase (UGM). Bioorganic
& Medicinal Chemistry Letters 2015,
25: 1995-7. |
|
 |
Kuppala R,
Mugunthan G, Tambat R, Patel N,
Nandanwar H, Bhutani KK and
Kartha KPR. Synthesis and
antibacterial activity of
ricinoleic acid glycosides. RSC
Advances 2016,
6: 3700-13. |
|
 |
Kumar R, Garg P, Bharatam PV. Shape-based virtual
screening, docking and molecular
dynamics simulations to identify
Mtb-ASADH inhibitors.J.
Biomol. Struct. Dyn.
2015,
33:
1082-93. |
|
 |
Abbat S, Jain V, Bharatam
PV. Origins of the specificity
of inhibitor P218 toward
wild-type and mutant PfDHFR:
A molecular dynamics analysis.J.
Biomol. Struct. Dyn.
2015,
33: 1913-28. |
|
 |
Dhaked DK,
Bharatam PV. DFT study on the
oxo transfer mechanism in
nitroethenediamine based
H2-receptor antagonists using
N-oxide reductase enzyme.
J. Bio. Inorg. Chem.
2015, 142: 84-91. |
|
 |
Kumar KA,
Kannaboina P, Dhaked DK,
Vishwakarma RA, Bharatam PV, Das
P. Cu-catalyzed N-arylation of
indazoles with boronic acids:
Synthesis of
pyrazolo-carbazolesvia
Pd-catalyzed oxidative cross-dehydrogenative
coupling. Org. Biomol.
Chem. 2015, 13: 1481-91. |
|
 |
Kumar CD, Sirisha
K, Dhaked DK, Lokesh P, Sarma
AVS, Bharatam PV.
Investigation of anion-pi
interactions involving thiophene
walls incorporated calix [4]
pyrroles. J.
Org. Chem. 2015, 80:
1746-53. |
|
 |
Gupta M, Jangra
H, Bharatam PV, Madan AK. Detour
Cum Distance Matrix Based
Topological Descriptors for QSAR/QSPR
Part-I: Development and
Evaluation. Lett. Drug
Design Disc. 2015,11:
844-63. |
|
 |
Baviskar AT,
Amrutkar SM, Trivedi N,
Chaudhary V, Nayak A, Guchhait
SK, Banerjee UC, Bharatam PV,
Kundu CN. Catalytic inhibition
of human topoisomerase IIa by
imidazopyridines: Switch in the
site ofinhibition from the ATP–
to the merbarone–binding domain.
ACS Med. Chem. Lett.
2015,
6:
481–5. |
|
 |
Bharate JB, Abbat
S, Sharma R, Bharatam PV,
Vishwakarma R, Bharate SB.
Cobalt (II) catalyzed C(sp)-H
bond functionalization of
alkynes with phenyl hydrazines:
A facile access to diaryl
1,2-diketones. Org. Biomol.
Chem. 2015, 13: 5235-42. |
|
 |
Sharma R, Abbat
S, Bharate JB, Bharate SB,
Bharatam PV, Vishwakarma R.
Ortho-quinone methides: TFA-mediated
generation in water and trapping
with lactams and styrenes.
Tetrahedron Letts.
2015, 56: 4057-9. |
|
 |
Ramakrishnan
A, Chourasiya S, Bharatam
PV. Azine or hydrazine? The
dilemma in amidinohydrazones.
RSC Advances 2015, 5:
55938-47. |
|
 |
Bharate JB, Abbat
S, Bharatam PV, Vishwakarma RA, Bharate SB.
CuBr catalyzed aerobic oxidative
coupling of 2-aminopyridines
with cinnamaldehydes: Direct
access to
3-formyl-2-phenyl-imidazo[1,2-a]pyridines.
Org. Biomol. Chem.
2015, 13:
7790-4. |
|
 |
Kusunuru AK,
Tatina M, Jaladanki CK, Bharatam
PV, Mukherjee D. Palladium
catalyzed diastereo selective
diarylation of glycals with aryl
boronic acids.Org. Letts.
2015, 17: 3742-5. |
|
 |
Rastogi GK, Abbat
S, Tiwari V, Fish MQ, Abrahams
S, Mosebi S, Killick M, Hewer
R, Papathanasopoulos MA,
Bharatam PV, Verma AK, Tandon V.
Molecular Docking, Synthesis and
Biological Evaluation of Novel
1,2-dihydroisoquinoline
derivatives as a next generation
HIV-1 integrase strand transfer
inhibitors (INSTI’s). ACS
Med. Chem. Letts. 2015,
6: 1065-70. |
|
 |
Patel M,
Saunthwal RK, Dhaked DK,
Bharatam PV, Verma AK. Nu-Addition
vs SNAr Study: Chemo-, Regio-
and Stereoselective Preferential
Hydrothiolation And
Hydroxylation of Haloarylalkynes
over S- and O-Arylation of Aryl
Halides. Asian
J. Org. Chem. 2016,
4, 894-898 |
|
 |
Kumar R, Garg P, Bharatam PV.
Pharmacoinformatics Analysis to
Identify Inhibitors of Mtb-ASADH. J.
Biomol. Struct. Dyn.
2015, DOI 10.1080/07391102.2015.1005137. |
|
 |
Chourasiya S,
Kathuria D, Singh S, Bharatam
PV, Sonavane V. An efficient
synthesis and biological
evaluation of novel azine
derivatives as quorum sensing
inhibitors. RSC Advances
2015,
5:
80027–38. |
|
 |
Abbat S, Dhaked
DK, Arfeen M, Bharatam PV.
Paal-Knorr synthesis of furan,
pyrrole and thiophene: A
mechanistic study using quantum
chemical methods. RSC
Advances 2015, 5:
88353-66. |
|
 |
Jaladanki CK, Taxak
N, Varikoti R, Bharatam PV.
Toxicity Originating from
Thiophene Containing Drugs:
Exploring the Mechanism using
Quantum Chemical Methods.
Chem. Res. Tox. 2015,
28: 2364–76. |
|
 |
Arfeen M, Patel
R, Khan T, Bharatam PV.
Molecular dynamics simulation of
GSK3b ATP competitive
inhibitors: Understanding the
factors contributing to
selectivity. J. Biomol.
Struct. Dyn. 2015, 33:
2578-83. |
|
 |
Chavan RB, Modi
SR, Bansal AK. Role of solid
carriers in pharmaceutical
performance of solid
supersaturable SEDDS of
celecoxib. International
Journal of Pharmaceutics
2015, 495 (1): 374-84. |
|
 |
Bhatt V, Shete G, Bansal AK.
Mechanism of generation of drug
nanocrystals in celecoxib:
mannitol nanocrystalline solid
dispersion. International
Journal of Pharmaceutics
2015, 495 (1): 132-9. |
|
 |
Sharma P, Modi
SR, Bansal AK. Co-processing as
a tool to improve aqueous
dispersibility of cellulose
ethers. Drug Development
and Industrial Pharmacy
2015, 41 (11): 1745-58. |
|
 |
Shete G, Modi SR,
Bansal AK. Effect of Mannitol on
Nucleation and Crystal Growth of
Amorphous Flavonoids:
Implications on the Formation of
Nanocrystalline Solid
Dispersion. Journal of
Pharmaceutical Sciences
2015, 104 (11): 3789-97. |
|
 |
Kumar D,
Thipparaboina R, Modi SR, Bansal
AK, Shastri NR. Effect of
surfactant concentration on
nifedipine crystal habit and its
related pharmaceutical
properties. Journal of
Crystal Growth 2015,
422: 44-51. |
|
 |
Sharma RJ, Gupta
RC, Bansal AK, Singh IP.
Metabolite Fingerprinting of
Eugenia jambolana Fruit Pulp
Extracts using NMR, HPLC-PDA-MS,
GC-MS, MALDI-TOF-MS and ESI-MS/MS
Spectrometry. Natural
Product Communications
2015, 10 (6): 969-76. |
|
 |
Sharma P, Modi
SR, Bansal AK. Co-processing of
hydroxypropyl methylcellulose (HPMC)
for improved aqueous
dispersibility.
International Journal of
Pharmaceutics 2015, 485
(1): 348-56. |
|
 |
Shete G, Pawar YB,
Thanki K, Jain S, Bansal AK.
Oral bioavailability and
pharmacodynamic activity of
hesperetin nanocrystals
generated using a novel
bottom-up technology.
Molecular Pharmaceutics
2015, 12 (4): 1158-70. |
|
 |
Munjal B, Bansal
AK. Counter-intuitive effect of
non-crystallizing sugars on the
crystallization of gemcitabine
HCl in frozen solutions.
International Journal of
Pharmaceutics 2015, 478
(1): 46-52. |
|
 |
Munjal B, Koradia
V, Boddu SHS, Bansal AK. Role of
Innovator Product
Characterization in Generic
Product Development.
Excipient applications in
formulation design and drug
delivery 2015, 521-38. |
|
 |
Kumar D,
Thipparaboina R, Modi SR, Bansal
AK, Shastri NR. Effect of HPMC
concentration on crystal habit
of nifedipine.
CrystEngComm 2015, 17
(7): 1615-24. |
|
 |
Sharma M, Akhtar
N, Sambhav K, Shete G, Bansal
AK, Sharma SS. Emerging
potential of citrus flavanones
as an antioxidant in diabetes
and its complications.
Current Topics In Medicinal
Chemistry 2015, 15 (2):
187-95. |
|
 |
Munjal B, Bansal
AK. Impact of Tert‐Butyl
Alcohol on Crystallization
Kinetics of Gemcitabine
Hydrochloride in Frozen Aqueous
Solutions. Journal Of
Pharmaceutical Sciences
2015, 104 (1): 87-97. |
|
 |
Patel J, Jagia M,
Bansal AK, Patel S.
Characterization and
Thermodynamic Relationship of
Three Polymorphs of a Xanthine
Oxidase Inhibitor, Febuxostat.
Journal Of Pharmaceutical
Sciences 2015, 104 (11):
3722-30. |
|
 |
Tarate B, Bansal
AK. Characterization of CoQ
10-lauric acid eutectic system.
Thermochimica Acta
2015, 605: 100-106. |
|
 |
Choudhary A,
Radhika M, Chatterjee A,
Banerjee UC, Singh IP.
Qualitative and quantitative
analysis of Potentilla
fulgens roots by NMR,
Matrix-assisted Laser Desorption/Ionisation
with Time-of-Flight MS,
Electrospray Ionisation MS/MS
and HPLC-UV. Phytochemical
Analysis 2015,
26:161–70. |
|
 |
Chauthe SK,
Mahajan S, Rachamala M, Tikoo K,
Singh IP. Synthesis and
evaluation of linear
furanocoumarins as potential
anti-breast and anti-prostate
cancer agents. Medicinal
Chemistry Research 2015,
24: 2476-84. |
|
 |
Saraf I,
Choudhary A, Sharma RJ, Dandi K,
Marsh KJ, Foley WJ, Singh IP.
Extraction of pinocembrin from
different species of
Eucalyptus leaves and its
quantitative analysis by qNMR
and HPTLC.
Natural
Product Communications
2015, 10: 379-82. |
|
 |
Choudhary A,
Kumar R, Srivastava RB,
Surapaneni SK, Tikoo K, Singh
IP. Isolation and
characterization of phenolic
compounds from Rhodiola
imbricata, a Trans-Himalyan
food crop having antioxidant and
anticancer potential.
Journal of Functional Foods
2015, 16:183-93. |
|
 |
Mittal AK,
Choudhary A, Tripathy D, Aili PK,
Ghanghoriya A, Chatterjee A,
Singh IP, Banerjee UC.
Bio-synthesis of
silver nanoparticles using
Potentilla fulgens ex wall.
Hook and its therapeutic
evaluation as anticancer and
antimicrobial agent.
Materials Science and
Engineering C. 2015, 53:
120-7. |
|
 |
Marsh KJ, Yin B,
Singh IP, Saraf I, Choudhary A,
Au J, Tucker DJ, Foley WJ.
From leaf metabolome to in
vivotesting:
Identifying antifeedant
compounds for ecological studies
of marsupial diets.
Journal of Chemical Ecology
2015, 41: 513-9. |
|
 |
Tripathy D,
Choudhary A, Banerjee UC, Singh
IP, Chatterjee A. Induction of
apoptosis and reduction of
endogenous glutathione level by
the ethyl-acetate soluble
fraction of the methanol extract
of the roots of
Potentilla
fulgens
in cancer cells. PLoS ONE
2015,
DOI:10.1371/journal.pone.0135890. |
|
 |
Singh IP and Choudhary
A. Piperine and Derivatives:
Trends in Structure-Activity
Relationships. Current
Topics in Medicinal Chemistry
2015, 15: 1722-34. |
|
 |
Devasari N, Dora CP, Singh C,
Paidi SR, Kumar V, Sobhia ME,
Suresh S. Inclusion complex of
erlotinib with sulfobutyl
ether-?-cyclodextrin:
Preparation, characterization,
in silico, in vitro and in vivo
evaluation. Carbohydrate
polymers 2015,
134:547-56. |
|
 |
Grover J, Bhatt N, Kumar V,
Patel NK, Gondaliya BJ, Sobhia
ME, Bhutani KK, Jachak SM. 2,
5-Diaryl-1, 3, 4-oxadiazoles as
selective COX-2 inhibitors and
anti-inflammatory agents.
RSC Advances 2015,
5(56):45535-44. |
|
 |
Kumar V, Sobhia ME. Molecular
Dynamics Assisted Mechanistic
Study of Isoniazid-Resistance
against Mycobacterium
tuberculosis InhA.
PloS one 2015,
10(12):e0144635. |
|
 |
Singh C, Koduri LSK, Kumar UA,
Bhatt TD, Kumar V, Sobhia ME,
Suresh S. Attenuation potential
of rifampicin?phospholipid
complex in murine hepatotoxicity
model. Journal of Drug
Delivery Science and Technology
2015, 30:225-31. |
|
 |
Iyer P, Bolla J, Kumar V, Gill
MS, Sobhia ME. In silico
identification of targets for a
novel scaffold,
2-thiazolylimino-5-benzylidin-thiazolidin-4-one.
Molecular diversity
2015. 19(4):855-70. |
|
 |
Grewal, B, Bhat J, Sobhia ME.
Molecular dynamics approach to
probe PKC?II?ligand interactions
and influence of crystal water
molecules on these interactions.
Expert opinion on
therapeutic targets
2015, 19(1):13-23 |
|
 |
Kumar V and Sobhia ME. Molecular
dynamics-based investigation of
InhA substrate binding loop for
diverse biological activity of
direct InhA inhibitors.
Journal of Bimolecular Structure
and Dynamics 2015.
(doi:10.1080/07391102.2015.111841)
(in press). |
 |
Devasari N, Dora CP, Singh C,
Paidi SR, Kumar V, Sobhia ME,
Suresh S. Inclusion complex of
erlotinib with sulfobutyl
ether-β-cyclodextrin:
Preparation, characterization,
in silico, in vitro and in vivo
evaluation. Carbohydrate
polymers 2015,
134:547-56. |
 |
Kumar V, Sobhia ME. Molecular
Dynamics Assisted Mechanistic
Study of Isoniazid-Resistance
against Mycobacterium
tuberculosis InhA. PLoS
ONE 2015,
10(12):e0144635. |
 |
Singh C, Koduri LSK, Kumar UA,
Bhatt TD, Kumar V, Sobhia ME,
Suresh S. Attenuation potential
of rifampicin–phospholipid
complex in murine hepatotoxicity
model. Journal of Drug
Delivery Science and Technology
2015, 30:225-31. |
 |
Iyer P, Bolla J, Kumar V, Gill
MS, Sobhia ME. In silico
identification of targets for a
novel scaffold,
2-thiazolylimino-5-benzylidin-thiazolidin-4-one.
Molecular Diversity
2015, 19(4):855-70. |
 |
Kumar V and Sobhia ME. Molecular
dynamics-based investigation of
InhA substrate binding loop for
diverse biological activity of
direct InhA inhibitors.
Journal of Bimolecular Structure
and Dynamics 2015,
(doi:10.1080/07391102.2015.1118410). |
|
 |
Guchhait SK and
Priyadarshani G. Pd-Catalyzed
Ag(I)-promoted C3-arylation of
pyrido[1,2‑a]pyrimidin-4-ones
with bromo/iodo-arenes.
J. Org. Chem. 2015,
80: 8482-88. |
|
 |
Guchhait SK and
Priyadarshani G. Synthesis of
2-arylpyridopyrimidinones,
6-aryluracils and tri- and
tetra-substituted conjugated
alkenes via Pd-catalyzed enolic
C–O bond activation-arylation.
J. Org. Chem.
2015, 80: 6342-49. |
|
 |
Chaudhary V, Das S, Guchhait SK
and Kundu C. Scaffold-hopping
and hybridization based design
and building block strategic
synthesis of pyridine-annulated
purines: discovery of novel
apoptotic anticancer agents.
RSC Adv.
2015,
5:
26051-60. |
|
 |
Chauhan AS, Rawat P, Malhotra H,
Sheokand N, Kumar M, Patidar A,
Chaudhary S, Jakhar P, Raje CI
and Raje M. Secreted
multifunctional
Glyceraldehyde-3-phosphate
dehydrogenase sequesters
lactoferrin and iron into cells
via a non-canonical pathway.
Scientific Reports
2015, 5:18465 doi:
10.1038/srep18465. |
|
 |
Agrawal AK, Urimi D, Harde H,
Kushwah V, Jain S. Folate
appended chitosan nanoparticles
augment the stability,
bioavailability and efficacy of
insulin in diabetic rats
following oral administration.
RSC Advances 2015,
5: 105179–93. |
|
 |
Jain S, Spandana
G, Agrawal AK, Kushwah V, Thanki
K. Enhanced antitumor efficacy
and reduced toxicity of
Docetaxel loaded Estradiol
functionalized stealth polymeric
nanoparticles.
Molecular
Pharmaceutics
2015, 12(11): 3871-84. |
|
 |
Sharma G, Beg S,
Thanki K, Katare OP, Jain S,
Kohli K, Singh B. Systematic
development of novel cationic
self-nanoemulsifying drug
delivery systems of Candesartan
Cilexetil with enhanced
biopharmaceutical performance.
RSC Advances
2015, 5: 71500-513. |
|
 |
Beg S, Sharma G,
Thanki K, Jain S, Katare OP,
Singh B. Positively charged
self-nanoemulsifying oily
formulations of Olmesartan
Medoxomil: Systematic
development, in vitro, ex
vivo and in vivo
evaluation. International
Journal of Pharmaceutics
2015, 493: 466-82. |
|
 |
Garg NK, Singh B,
Sharma G, Kushwah V, Tyagi RK,
Jain S, Katare OP. Development
and characterization of single
step self assembled lipid
polymer hybrid nanoparticles for
effective delivery of
Methotrexate. RSC Advances
2015, 5: 62989-99. |
|
 |
Harde H, Agrawal
AK, Jain S. Tetanus
toxoid loaded layer-by-layer
nanoassemblies for efficient
systemic, mucosal and cellular
immunostimulatory response
following oral administration.
Drug Delivery and
Translational Research
2015, 5(5): 498-510. |
|
 |
Jain S, Kambam S,
Thanki K, Jain AK. Cyclosporine
A loaded self-nanoemulsifying
drug delivery system (SNEDDS):
Implication of functional
excipient based co-encapsulation
strategy on oral bioavailability
and nephrotoxicity. RSC
Advances 2015, 5:
49633-42. |
|
 |
Jain S, Bhankur
N, Swarnakar NK, Thanki K.
Phytantriol based “Stealth”
lyotropic liquid crystalline
nanoparticles for improved
antitumor efficacy and reduced
toxicity of Docetaxel.
Pharmaceutical Research
2015, 23(10): 3282-92. |
|
 |
Harde H, Agrawal
AK, Katariya M, Kale D,
Jain S.
Development of topical Adapalene-solid
lipid nanoparticles loaded gel
with enhanced efficacy and
improved skin tolerability.
RSC Advances
2015, 5: 43917–29. |
|
 |
Arora S, Haghi M,
Loo CY, Traini D, Young PM,
Jain S. Development of an
inhaled controlled release
Voriconazole dry powder
formulation for the treatment of
respiratory fungal infection.
Molecular
Pharmaceutics
2015, 12(6):
2001-9. |
|
 |
Jain S,
Kumar S, Agrawal AK, Thanki K,
Banerjee UC.
Hyaluronic
acid-PEI-cyclodextrin polyplexes:
Implications on in vitro and in
vivo transfection efficiency and
toxicity.
RSC Advances
2015, 5: 41144–54. |
|
 |
Arora S, Mahajan
RR, Kushwah V, Baradia D, Misra
AN, Jain S. Development of
Voriconazole loaded large porous
particles for inhalation
delivery: Effect of surface
forces on aerosolisation
performance, assessment of in
vitro safety potential and
uptake by macrophages.
RSC Advances
2015, 5: 38030–43. |
|
 |
Harde H,
Siddhapura K, Agrawal AK, Jain
S.
Divalent toxoids loaded stable
Chitosan-glucomannan
nanoassemblies for efficient
systemic, mucosal and cellular
immunostimulatory response
following oral administration.
International Journal of
Pharmaceutics 2015,
487(1-2): 292-304. |
|
 |
Harde H,
Siddhapura K, Agrawal AK, Jain
S.
Development of dual toxoids
loaded layersomes for complete
immuno-stimulatory response
following peroral
administration.
Nanomedicine
(London)
2015, 10(7):
1077-91. |
|
 |
Rai VK, Mishra N,
Agrawal AK, Jain S, Yadav NP.
Novel drug delivery system: an
immense hope for diabetics.
Drug Delivery 2015,
25: 1-20. |
|
 |
Kapoor R, Harde
H, Jain S, Panda AK, Panda BP.
Downstream processing,
formulation development and
antithrombotic evaluation of
microbial Nattokinase.
Journal of
Biomedical Nanotechnology
2015, 11: 1213-24. |
|
 |
Harde H, Agrawal
AK, Jain S. Tetanus toxoid
loaded glucomannosylated
Chitosan based nanohoming
vaccine adjuvant with improved
oral stability and
immunostimulatory response.
Pharmaceutical Research
2015, 32: 122-34. |
|
 |
Harde H, Agrawal
AK, Jain S.
Development of
stabilized mannosylated chitosan
nanoparticles for oral delivery:
Demonstration of immunization
using BSA as model antigen.
Nanomedicine
(London)
2015, 9(16):
2511-29. |
|
 |
Dinesh N, Soumya N and Singh S.
Antileishmanial effect of mevastatin is due to interference
with sterol metabolism.
Parasitol Res.
2015, 114(10):3873-83. |
|
 |
Soumya N, Kumar IS, Shivaprasad S, Gorakh LN,
Dinesh N, Swamy KK and Singh S. AMP-acetyl CoA synthetase
from Leishmania donovani: identification and functional
analysis of 'PX4GK' motif.
Int. J Biol Macromol.
2015, 75:364-72. |
|
 |
Borkar RM, Bhandi
MM, Dubey AP, Nandekar PP,
Sangamwar AT,
Baberjee SK,
Srinivas R. Plasma protein
binding, pharmacokinetics,
tissue distribution, and CYP450
biotransformation studies of
fidarestat by ultra high
performance liquid
chromatography-high resolution
mass spectrometry. J Pharm
Biomed Anal. 2015, 102:
386-99. |
|
 |
Patel SR, Gangwal R, Sangamwar
AT, Jain R. Synthesis,
biological evaluation and 3D
QSAR study of 2,4-disubstituted
quinolines as anti-tuberculosis
agents. Eur J Med Chem. 2015,
26(93): 511-22. |
|
 |
Mahindra A, Gangwal RP, Bansal
S, Goldfarb NE, Dunn BM,
Sangamwar AT and Jain
R.Antiplasmodial activity of
short peptide-based compounds.
RSC Adv. 2015, 5:
22674-84. |
|
 |
Patel PN, Borkar RM, Kalariya
PD, Gangwal RP, Sangamwar AT,
Gananadhamu S and Ragampeta S.
Characterization of degradation
products of Ivabradine by
LC-HR-MS/MS: a typical case of
exhibition of different
degradation behaviour in HCl and
H2SO4 acid hydrolysis. J
Mass Spectro 2015, 50(2):
344–53. |
|
 |
Gangwal RP, Damre MV, Das NR,
Dhoke GV, Bhadauriya A, Varikoti
RA, Sharma SS, Sangamwar AT.
Structure based virtual
screening to identify selective
phosphodiesterase 4B inhibitors
J Mol Graph Model.
2015, 57: 89-98. |
|
 |
Jena SK, Sarsija S, Sangamwar
AT. Modulation of tamoxifen
induced hepatotoxicity by
tamoxifen-phospholipid complex.
J Pharm Pharmacol
2015, Apr 23. |
|
 |
Dara A, Sangamwar AT. Technology
Whitespaces India Should Focus:
A Comparative Anticancer Patent
Rational Analysis of Indian and
International Public Funded
Universities. Recent Pat
Anticancer Drug Discov.
2015, 10(2): 163-9. |
|
 |
Chauhan PS, Tripathi SP,
Sangamwar AT, Puri N, Sharma P,
Gupta N. Cloning, molecular
modelling, and docking analysis
of alkali-thermostable β-mannanase
from Bacillus nealsonii PN-11.
ApplMicrobiolBiotechnol
2015, 99(21): 8917-25. |
|
 |
Patel NK, Bairwa K, Gangwal R,
Jaiswal G, Jachak SM, Abhay T
Sangamwar, Bhutani KK.
2’-hydroxy flavanone derivatives
as inhibitors of
pro-inflammatory mediators:
Experimental and molecule
docking studies. Biorg and
Med Chem Letters 2015,
25 (9): 1952-5. |
|
 |
Meena CL, Ingole S, Rajpoot S,
Thakur A, Nandekar PP, Sangamwar
AT, Sharma SS, Jain R. Discovery
of a low affinity thyrotropin
releasing hormone (TRH) like
peptide that exhibits potent
inhibition of scopolamine
induced memory impairment in
mice. RSC Advances
2015, 5: 56872-84. |
|
 |
Dara Ajay, Rahul P Gangwal,
Abhay T Sangamwar. IPAT: A
freely accessible software tool
for analysing multiple patent
documents with inbuilt landscape
visualizer. Pharmaceutical
Patent Analyst 2015,
4(5): 377-86. |
|
 |
Avasathi V, Pawar H, Dora CP,
Bansod P, Gill MS and Suresh S.
A novel nanogel formulation of
Methotrexate for topical
treatment of psoriasis:
optimization, in vitro and in
vivo evaluation. Pharm Dev
Technol 2015, 1-9. |
|
 |
Jain M, Burman RP, Negi VS,
Jhamb SS, Mital A and Gill MS.
Synthesis and Biological
Evaluation of
2-thiazolylimino-5-arylidene-4-
thiazolidinone Derivatives as
Potent Antimycobacterial Agents.
Anti-Infective Agents 2015,
13(2): 105-13. |
|
 |
Laha JK, Sharma
S, Dayal N. Palladium-Catalyzed
Regio- and Chemoselective
Reactions of 2-Bromobenzyl
Bromides: Expanding the Scope
for the Synthesis of Biaryls
Fused to a Seven-Membered Sultam. Eur.
J. Org. Chem. 2015,
7885-91. |
|
 |
Laha JK, Jethava KP, Patel S.
Scope of Successive C-H
Functionalizations of the Methyl
Group in 3-Picolines:
Intramolecular Carbonylation of
Arenes to the Metal-free
Synthesis of 4-Azafluorenones,
Org. Lett. 2015,
17: 5890-3. |
|
 |
Laha JK, Tummalapalli KSS, Nair,
A, Patel N. Sulfate Radical
Anion (SO4˙ˉ) Mediated C(sp3)-H
Nitrogenation/Oxygenation in
N-Aryl Benzylic Amines Expanded
the Scope for the Synthesis of
Benzamidine/oxazine Heterocycles. J.
Org. Chem. 2015, 80:
11351-59. |
|
 |
Laha JK, Dayal N. A Tandem
Approach to Functionalized
Carbazoles from Indoles via Two
Successive Regioselective
Oxidative Heck Reactions
Followed by Thermal
Electrocyclization. Org.
Lett. 2015, 17: 4742–45. |
|
 |
Laha
JK,
Dayal
N,
Jethava
KP,
Prajapati
DV. Access to Biaryl
Sulfonamides by
Palladium-Catalyzed
Intramolecular Oxidative
Coupling and Subsequent
Nucleophilic Ring Opening of
Heterobiaryl Sultams with
Amines. Org. Lett.
2015, 17: 1296–9. |
|
|
|
2014 |
|
 |
Karmase A, Prasanna K, S
Rasabattula S and Bhutani KK.
Quantification and comparison of
extraction methods for alkaloids
in Aegle marmelos leaves by HPLC.
Natural Products
Communication 2014,
9: 981-83. |
 |
Bhutani KK (Guest Editor),
Biotechnology Volume 7: Drug
Discovery, Studium Press
LLC, U.S.A., 1-566. |
 |
Baboota RK, Murtaza N, Jagtap S,
Singh DP, Karmase A, Kaur J,
Bhutani KK, Boparai RK,
Premkumar LS, Kondepudi KK and
Bishnoi M. Capsaicin-induced
transcriptional changes in
hypothalamus and alterations in
gut microbial count in high fat
diet fed mice. Journal of
Nutritional Biochemistry
2014, 25: 893-902. |
 |
Murtaza N, Baboota R, Jagtap S,
Singh D, Khare P, Sarma S,
Koteswaraiah P, Alagesan S,
Chandra TS, Bhutani KK, Boparai
R, Bishnoi M and Kondepudi KK.
Finger millet bran consumption
ameliorated obesity induced
oxidative stress, inflammation
and gut microbial derangements
in high fat diet fed mice.
British Journal of Nutrition
2014, 112:1447-58. |
 |
Lunagariya NA, Patel NK, Jagtap
SC and Bhutani KK. Inhibitors of
pancreatic lipase: State of the
art and clinical perspectives.
EXCLI Journal
2014, 13: 897-921. |
 |
Patel NK and Bhutani KK.
Suppressive effects of Mimosa
pudica (L.) constituents on the
production of LPS-induced
pro-inflammatory mediators.
EXCLI Journal 2014,
13: 1011-21. |
 |
Patel NK and Bhutani KK.
Pinostrobin and Cajanus lactone
isolated from Cajanus cajan (L.)
leaves inhibits TNF-α and IL-1β
production: In vitro and in vivo
experimentation.
Phytomedicine 2014,
21: 946-53. |
 |
Patel NK, Pulipaka S, Dubey SP
and Bhutani KK. Pro-inflammatory
cytokines and nitric oxide
inhibitory constituents from
Cassia occidentalis(L.) roots.
Natural Product
Communications 2014,
9: 661-64. |
 |
Kumar H, Pandey PK, Doiphode VV,
Vir S, Bhutani KK, Patole MS and
Shouche YS. Microbial Community
Structure at Different
Fermentation Stages of
Kutajarista, a Herbal
Formulation. Indian
Journal of Microbiol
(Jan–Mar 2013), 53(1): 11-17. |
 |
Bhandari P, Patel NK, Gangwal
RP, Sangamwar AT and Bhutani KK.
Oleanolic acid analogs as NO,
TNF-α and IL-1β inhibitors:
Synthesis, biological evaluation
and docking studies.
Bioorganic & Medicinal Chemistry
Letters 2014,
24(17): 4114-19. |
 |
Bhandari P, Patel NK and Bhutani
KK. Synthesis of new
heterocyclic lupeol derivatives
as nitric oxide and
pro-inflammatory cytokine
inhibitors. Bioorganic and
Medicinal Chemistry Letters
2014, 24(15): 3596-99. |
 |
Patel NK, Ramandeep and Bhutani
KK. Activity-guided
Fractionation of Ipomea
fistulosa leaves for
Proinflammatory Cytokines and
Nitric Oxide Inhibitory
Constituents. Natural
Product Communications
2014, 9:1749-50. |
 |
Natsume Y, Patel NK, Tripathi
SM, Nose M, Kyuma T and Bhutani
KK. Kalyanka Ghrta: an example
of intertextuality among The
Bower Manuscript, Charak samhita,
Sushruta samhita, Astangahrdayam
samhita and Ayurvedic Formulary
of India (AFI). Indian
Journal of Traditional Knowledge
2014, (accepted). |
 |
Jhajra S, Bhatia S, Bharatam PV
and Singh S. Explanation Through
Density Functional Theory of the
Unanticipated Loss of CO2
and Differences in Mass
Fragmentation Profiles of
Ritonavir and Its rCYP3A4
Mediated Metabolites.
Journal of Mass Spectrometry
2014, 49(6):452–67. |
 |
Kurmi M, Kumar S, Singh B and
Singh S. Implementation of
Design of Experiments for
Optimization of Forced
Degradation Conditions and
Development of a
Stability-Indicating Method for
Furosemide. Journal of
Pharmaceutical and Biomedical
Analysis 2014, 96:
135–43. |
 |
Narayanam M and Singh S.
Characterization of Stress
Degradation Products of
Fosinopril by Using LC-MS/TOF,
MSn and On-line H/D
Exchange. Journal of
Pharmaceutical and Biomedical
Analysis 2014,
92: 135–43. |
 |
Varkhede NR, Jhajra S, Ahire DS
and Singh S.
Metabolite Identification
Studies on Amiodarone in In
Vitro (Rat Liver Microsomes, Rat
And Human Liver S9 Fractions)
and In Vivo (Rat Feces, Urine,
Plasma) Matrices by Using LC-HRMS
and LC-MSn:
Characterization of Diquinone
Metabolite Supposedly
Responsible for the Drug’s
Hepatotoxicity.
Rapid Communications in Mass
Spectrometry 2014,
28 (4):
311-31. |
 |
Handa T, Singh IP and Singh S.
Characterization of a New
Degradation Product of
Nifedipine Catalyzed by Atenolol:
A Typical Case of Alteration of
Degradation Pathway of One Drug
by Another.
Journal of Pharmaceutical and
Biomedical
Analysis
2014,
89: 6–17. |
 |
Bhutani H, Kurmi M, Singh S, Beg
S and Singh B. Quality by Design
in Analytical Sciences: An
Overview. Pharmatimes
2014, 46(8): 71-75. |
 |
Jhajra
S,
Prasad B,
Shah J and
Singh S. High-resolution
MS for drug metabolite
identification,
In:
Applications of High-Resolution
Mass Spectrometry in Drug
Discovery and Development,
Future Science
Ltd.,
London N3 1QB, UK,
2014, Pages 22-40,
eBook ISBN: 978-1-909453-55-5. |
 |
Jindal K, Narayanam M and
Singh S. Pollution of Aqueous
Matrices with Pharmaceuticals.
In: Water and Health, PP
Singh and VP Sharma (Eds.),
Chapter 21, Springer-Cerlag,
India, 2014 pp.
355-373 (ISBN: 978-81-322-1028-3
(Print) 978-81-322-1029-0
(online). |
 |
Banoth
L,
Pujala
B,
Chakraborti
AK
and
Banerjee
UC.
Development and Validation of
HPLC Method for the Resolution
of Derivatives of
1_Bromo_3_Chloro_2_Propanol: a
Novel Chiral Building Block for
the Synthesis of
Pharmaceutically Important
Compounds.
Journal of Analytical
Chemistry 2014,
69: 1206–13. |
 |
Meena
VS,
Banoth
L and
Banerjee
UC.
Demostration of redox potential
of Metschnikowia koreensis for
stereoinversion of secondary
alcohols/1,2-diols.
BioMed Research
International
2014,
5: 2014. |
 |
Banoth
L,
Chandarrao
B,
Pujala
B,
Chakraborti
AK
and Banerjee
UC.
New and Efficient Chemical and
First Chemo-enzymatic Synthesis
of (RS)-, (R)-,
and (S)-Bunitrolol.
Synthesis 2014,
46(4): 479-88. |
 |
Mittal
AK,
Bhaumik
J,
Kumar
S
and Banerjee
UC.
Biosynthesis of silver
nanoparticles: elucidation of
prospective mechanism and
therapeutic potential.
Journal of Colloid and
Interface Science
2014,
415(1):39-47. |
 |
Pai
O,
Banoth
L,
Ghosh
S,
Chisti
Y and
Banerjee
UC.
Biotransformation of
3-cyanopyridine to nicotinic
acid by whole cells of
recombinant
Escherichia coli.
Process Biochemistry
2014, 49: 655–59. |
 |
Banoth
L and
Banerjee
UC.
New Chemical and
Chemo-enzymatic Synthesis of
(RS)-, (R)-, and (S)-Esmolol.
Arabian Journal of
Chemistry
(accepted
2014),
doi:10.1016/j.arabjc.2014.03.011. |
 |
Seth
K, Garg
SK,
Kumar
R,
Purohit
P, Meena
VS,
Goyal
R,
Banerjee
UC
and
Chakraborti
AK.
2-(2-Arylphenyl)benzoxazole As a
Novel Anti-Inflammatory
Scaffold: Synthesis and
Biological Evaluation.
ACS Medicinal Chemistry
Letters 2014,
5(5): 512-16. |
 |
Mittal
AK,
Kumar
S
and Banerjee
UC.
Quercetin and gallic acid
mediated synthesis of bimetallic
(Ag-Se) nanoparticles and their
antitumor and antimicrobial
potential.
Journal of Colloid and
Interface Science 2014,
431: 194-99. |
 |
Ghosh
S,
Pawar
H,
Pai
O
and Banerjee
UC.
Microbial
transformation of quinic acid to
shikimic acid by
Bacillus
megaterium.
Bioresources
and Bioprocessing
2014,1: 1-6. |
 |
Ghoshal
G,
Banerjee
UC
and Shivhare
US.
Xylanase
Production by Penicillium
citrinum in Laboratory Scale
Stirred Tank Reactor.
Chemical
& Biochemical Engineering
Quarterly
2014,
28(3):ISSN
No-1846-5153. |
 |
Ghoshal
G,
Banerjee
UC
and Shivhare
US.
Isolation, Screening and
Optimization of Xylanase
Production in Submerged
Fermentation Using P.citrinum.,
Journal of
Scientific & Industrial Research
2014
(accepted). |
 |
Kaler A, Mittal
AK, Katariya M, Harde H, Agrawal
AK, Jain S and Banerjee UC.
An investigation of in vivo
wound healing activity of
biologically synthesized silver
nanoparticles. Journal of
Nanoparticle Research
2014, 16: 2605. |
 |
Sav
A,
Mittal
A,
Thorat
A,
Dubey
S
and Banerjee
UC.
A comparative study on the
production of
Polyhydroxyalkanoate (PHA) by
three different Pseudomonas sp.
International Journal of
Current Microbiology and Applied
Sciences 2014,
3(10): 409-18. |
 |
Kumar V, Giri S.K, Paloth V and
Kartha KPR. Synthesis of
cross-linked glycopeptides and
ureas by a mechanochemical,
solvent-free reaction and
determination of their
structural properties by TEM and
X-ray crystallography,
ChemPlusChem 2014,
79:
1605-1613. |
 |
Kumar V, Taxak N, Jangir R,
Bharatam PV and Kartha KPR.
In(III) Triflate-mediated
solvent-free synthesis and
activation of thioglycosides by
ball milling and structural
analysis of long chain alkyl
thioglycosides by TEM and
quantum chemical methods,
J. Org Chem. 2014, 79: 3427-39. |
 |
Kumar V, Narender N and Kartha
KPR. In(III) triflate-catalyzed
detritylation and glycosylation,
Carbohydr. Res.
2014, 397: 18-26. |
 |
Singh JN, Rathej
M and Sharma SS.
Diabetic-induced increased
sodium channel activity
attenuated by tetracaine in
sensory neurons in vitro.
Biochem Biophys Res Comm
2014,
453(3): 296-301. |
 |
Das NR, Gangwal
RP, Damre MV, Sangamwar AT
and
Sharma SS.
A PPAR-β/δ
agonist is neuroprotective and
decreases cognitive impairment
in a rodent model of Parkinson’s
disease. Current
Neurovascular Research
2014, 11(2): 114-24. |
 |
Uppalapati D, Das NR, Gangwal
RP, Damre MV, Sangamwar AT
and
Sharma SS. Neuroprotective
Potential of Peroxisome
Proliferator Activated
Receptor-𝛼
Agonist
in Cognitive Impairment in
Parkinson’s Disease: Behavioral,
Biochemical, and PBPK Profile.
PPAR Research
2014: 2014,
doi:10.1155/2014/753587. |
 |
Gangwal RP, Das
NR, Thanki K, Damre MV,
Dhoke GV, Sharma SS, Jain S and
Sangamwar AT.
Identification of
p38 MAP kinase inhibitors by
Pharmacophore based virtual
screening. Journal of
Molecular Graphics and Modelling
2014, 49: 18-24. |
 |
Jangra A,
Datusalia A, and Sharma SS.
Reversal of neurobehavioral and
neurochemical
alterations in STZ-induced
diabetic rats by
FeTMPyP, a peroxynitrite
decomposition
catalyst and
1,5-Isoquinolinediol a poly(ADP-ribose)
polymerase
inhibitor. Neurological
Research 2014,
36(7): 619-26. |
 |
Dhaked DK and Bharatam PV.
Conformational and zwitterionic
preferences of N-amidinoglycine:
The effect of microsolvation and
metal ion addition. RSC
Advances 2014, 4:
4533-44. |
 |
Mudududdla R, Sharma R, Abbat S
and Bharatam PV, Vishwakarma RA,
Bharate SB. Synthesis of
2-phenyl naphthalenes from
styryl-2-methoxybenzenes.
Chem. Commun. 2014,
12076-79. |
 |
Kaur R, Ramesh M, Bharatam PV
and Kishore R. Self-Association
Behaviour of a Novel Non-Proteinogenic
β-Strand- Mimic in an Organic
Solvent. J. Phys. Chem. B
2014, 118: 9199-9208. |
 |
Madan J, Gundala SR, Kasetti Y,
Bharatam, Aneja R, Katyal A and
Jain UK. Enhanced Noscapine
Delivery Using Estrogen-Receptor
Targeted Nanoparticles for
Breast Cancer Therapy.
Anticancer Drugs 2014,
25(6): 704-16. |
 |
Bharatam PV, Arfeen M, Abbat S,
Patel DS and Taxak N. Quantum
chemical studies on the
cyclisation of anti-malarial
Proguanil. J. Comput.
Chem. 2014, 35: 2047-55. |
 |
Sanghai N, Jain V, Preet R,
Kandekar S, Das S, Trivedi N,
Mohapatra P, Priyadarshani G,
Kashyap M, Das D, Sathapathy SR,
Siddhardh S, Guchhait SK, Kundu
CN and Bharatam PV.
Combretastatin A-4 Inspired
Novel
2-Aryl-3-arylamino-imidazo-pyridine/pyrazines
as Tubulin Polymerization
Inhibitors, Antimitotic, and
Anticancer Agents. Med.
Chem. Comm. 2014, 5:
766-82. |
 |
DhakedDK and Bharatam PV. On the
stability of zwitter ions of
Pyridine sulfonylureas : The
Effect of isosterim, acidity and
microsolvation. J. Phys.
Chem. A 2014, 118:
187-96. |
 |
Bhatia S and Bharatam PV.
Possibility of existence of
Donon-acceptor interactions in
medicinally important
bis(azole)amine derivatives.
J. Org. Chem. 2014, 79:
4852–62. |
 |
Gupta M, Jangra H, Bharatam PV
and Madan AK. Relative eccentric
distance sum/product indices for
QSAR/QSPR: Development,
evaluation and application.
ACS Comb. Sci. 2014, 16:
101-12. |
 |
Singh M, Jangra H, Bharatam PV
and Madan AK. Detour
Matrix-based Adjacent Path
Eccentric Distance Sum Indices
for QSAR/QSPR Part I:
Development and Evaluation.
Int. J. Comput. Biol. Drug
Design 2014, 7: 295-318. |
 |
Bharatam PV, Adane L, Bhagat S,
Arfeen M, Bhatia S, Sirawaraporn
R, Sirawaraporn W and
Chakraborti AK. Design and
synthesis of guanylthiourea
derivatives as potential
inhibitors of Plasmodium
falciparum Dihydrofolate
Reductase enzyme. Bioorg.
Med. Chem. Letts. 2014,
24: 613-17. |
 |
Ramesh M and Bharatam PV.
Importance of hydrophobic
parameters in identifying
appropriate pose of CYP
substrate in cytochromes.
Eur. J. Med. Chem. 2014,
71: 15-23. |
 |
Mahindra A, Bagra N, Wangoo N,
Khan SI, Jacob MR and Jain R.
Discovery of short peptides
exhibiting high potency against
Cryptococcus neoformans.
ACS Med. Chem. Lett.
2014, 5: 315-20. |
 |
Mahindra A, Sharma KK, Rathore
D, Khan SI, Jacob MR and Jain R.
Synthesis and antimicrobial
activities of His(2-aryl)-Arg
and Trp-His(2-aryl) classes of
dipeptidomimetics.
Med. Chem. Commun. 2014,
5: 671-76. |
 |
Mahindra R
and
Jain R.
Regiocontrolled
palladium-catalyzed and
copper-mediated C-H bond
functionalization of protected
L-histidine.
Org. Biomol. Chem. 2014,
12: 3792-96. |
 |
Mahindra A, Bagra N, Wangoo N,
Jain R, Khan SI, Jacob MR and
Jain R. Synthetically modified
L-histidine-rich
peptidomimetics exhibit potent
activity against
Cryptococcus neoformans.
Bioorg. Med. Chem. Lett.
2014, 24: 3150-54. |
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Bagul
P, Khomane K, Kesharwani S,
Pragyan P, Nandekar P, Meena
C, Bansal A, Jain R, Tikkoo
K
and Sangamwar A. Intestinal
transport of TRH analogues
through PepT1: The role of in
silico and in vitro modelling.
J. Mol. Recognit.
2014,
27(10): 609-17. |
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Patel
S, Gangwal R, Sangamwar AT
and Jain
R. Synthesis, biological
evaluation and 3D-QSAR study of hydrazide, semicarbazide and
thiosemicarbazide derivatives of
4-(1-adamantan-1-yl)quinoline as
anti-tuberculosis agents.
Eur.
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85: 255-67. |
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Mahindra A, Patel N, Bagra N and
Jain R. Solvent-free peptide
synthesis assisted by microwave
irradiation: environmentally
benign synthesis of bioactive
peptides.
RSC Adv.
2014, 4: 3065-69. |
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Tiwari P, Ahlawat
R and Gupta G. Pharmacoepidemiological
profiling of acute
gastroenteritis patients at a
paediatric outpatient setting.
Ind J Hosp Pharm
2014, 51: 116-20. |
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Ahlawat R, Gupta
G and Tiwari P. Complementary
medicine causing severe
side-effects in a child - an
overlooked cause of weight
loss?. Int J Pharm Sci Res
2014, 5: 478-9. |
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Tiwari P, Ahlawat
R and Gupta G. Prescription
practice in patients of upper
respiratory tract infection at a
pediatric outpatient clinic in
Punjab. Ind J Pharm Pract
2014, 7:1-7. |
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Ahlawat R, Tiwari
P and Gupta G. Assessment of
prescribing at a private
pediatric outpatient setting in
northern India. Asian J
Clin Pediatr Neonatol
2014, 2: 23-7. |
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Bansal D, Mangla
S, Undela K, Gudala K, D'Cruz S,
Sachdev A and Tiwari P. Measurement
of adult antimicrobial drug use
in tertiary care hospital using
defined daily dose and days of
therapy. Indian J Pharm
Sci. 2014, 76: 211-17. |
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GBN Sireesha,
Tiwari P, Gombar S, D'Cruz S
and Sachdev A. Antimicrobial
utilisation study in
multidisciplinary intensive care
units of a public tertiary care
hospital. J Pharmacol
Pharmacother 2014, 5:
252. |
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Undela
K, Bansal D, D'Cruz S, Sachdev
A and Tiwari P. Prevalence and
determinants of use of
potentially inappropriate
medications in elderly
inpatients: a prospective study
in a tertiary healthcare
setting. Geriatr Gerontol
Intl. 2014, 14: 251-8. |
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Patil SP,
Modi SR and
Bansal AK.
Generation of 1:1 Carbamazepine:
Nicotinamide cocrystals by spray
drying. European Journal
of Pharmaceutical Sciences
2014, 62: 251-57. |
 |
Khomane K and
Bansal AK. Differential
compaction behaviour of roller
compacted granules of
clopidogrel bisulphate
polymorphs. International
Journal of Pharmaceutics
2014, 472(1-2): 288-95. |
 |
Kumar, Mehul,
Munjal B and Bansal AK.
Differential effect of buffering
agents on the crystallization of
gemcitabine hydrochloride in
frozen solutions.
International Journal of
Pharmaceutics
2014, 471(1-2): 56-64. |
 |
Shete
G, Kuncham S, Puri V, Gangwal
R, Sangamwar A and Bansal A.
Effect of different states of
‘sorbed’ water on amorphous celecoxib.
Journal of
Pharmaceutical Sciences
2014,
103: 2033-41. |
 |
Nanakwani K, Modi
SR, Kumar L and Bansal AK. Role
of thermodynamic, kinetic and
structural factors in the
recrystallization behavior of
amorphous erythromycin salts.
Thermochimica Acta 2014,
582: 77-85. |
 |
Bagul P, Khomane
K and Bansal AK. Investigating
permeability related hurdles in
oral delivery of
11-keto-β-boswellic acid.
International Journal of
Pharmaceutics 2014,
464(1-2): 104-110. |
 |
Kuncham, S, Shete
G and Bansal AK. Quantification
of clarithromycin polymorphs in
presence of tablet excipients.
Journal of Excipients and
Food Chemicals 2014,
5(1): 65-78. |
 |
Tarate B, Chavan
R and Bansal AK. Oral Solid
Self-emulsifying Formulations: A
Patent Review. Recent
Patents on Drug Delivery &
Formulation 2014, 8(2):
126-43. |
 |
Modi S, Khomane
KS and Bansal AK.
Impact of
differential surface molecular
environment on the
interparticulate bonding
strength of celecoxib crystal
habits. International Journal of
Pharmaceutics
2014,
460(1-2):
189-195. |
 |
Jain HK, Kailas K
and Bansal AK. Implication of
microstructure on the mechanical
behaviour of an aspirin–paracetamol
eutectic mixture.
Crystal
Engineering Communication
2014,
16: 8471-78. |
 |
Dani P, Puri V
and Bansal AK. Solubility
advantage from amorphous
etoricoxib solid dispersions.
Drug Development and
Industrial Pharmacy
2014, 40(1): 92-101. |
 |
Shete G and
Bansal AK. Molecular relaxation
behavior and isothermal
crystallization above
glass-transition temperature of
amorphous hesperetin.
Journal of Pharmaceutical
Sciences 2014,
103(1): 167-78. |
 |
Shete G, Jain H,
Punj D, Prajapat H, Akotiya P,
Bansal AK. Stabilizers used in
nanocrystal based drug delivery
systems. Journal of
Excipients and Food Chemicals
2014, 5(4): 184-209. |
 |
Bansal AK.
Excipients used in nano-technology
assisted drug delivery systems.
Journal of Excipients and
Food Chemicals 2014, 5(4): 173-76. |
 |
Bulani Y, Sambhav K, Akhtar N,
Shete G, Bansal AK and Sharma
SS. Effect of Nanocrystalline
Solid Dispersion Formulation of
Hesperetin in Diabetic
Cardiomyopathy. Indian
Journal of Pharmacology
2014, 46: S30-S30 |
 |
Sheokand S, Modi
SR and Bansal AK. Dynamic Vapor
Sorption as a Tool for
Characterization and
Quantification of Amorphous
Content in Predominantly
Crystalline Materials.
Journal of Pharmaceutical
Sciences 2014, 103(11):
3364-76. |
 |
Modi SR,
Dantuluri AKR, Perumalla SR, Sun
CC and Bansal AK. Effect of crystal
habit on intrinsic dissolution
behavior of celecoxib due to
differential wettability.
Crystal Growth & Design
2014, 14(10): 5283-92. |
 |
Kumar GS,
Kulkarni A, Khurana A, Kaur J
and
Tikoo K.
Selenium nanoparticles involve
HSP-70 and SIRT1 in preventing
the progression of type 1
diabetic nephropathy.
ChemBiol Interact. 2014,
223C:
125-33. |
 |
Kulkarni A, Kumar
GS, Kaur J
and
Tikoo K. A comparative study of
the toxicological aspects of
vanadium pentoxide and vanadium
oxide nanoparticles.
InhalToxicol. 2014,
26(13):
772-88. |
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Bairwa K and Jachak SM.
Anti-inflammatory potential of a
lipid based formulation of
rotenoid rich fraction prepared
from Boerhaavia diffusa
L. Pharmaceutical Biology
2014, 53: 1231-38. |
 |
Grover J, Kumar V, Singh V,
Bairwa K, Sobhia ME and Jachak
SM. Synthesis, biological
evaluation, molecular docking
and theoretical evaluation of
ADMET properties of nepodin and
chrysophanol derivatives as
potential cyclooxygenase (COX-1,
COX-2) inhibitors. Eur J
Med Chem. 2014,
80: 47-56. |
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Bairwa K, Srivastava A, Jachak
SM. Quantitative analysis of
boeravinones in the roots of
Boerhaavia diffusa by UPLC-PDA.
Phytochemical Analysis
2014, 25: 415-20. |
 |
Grover J, Roy SK, Jachak SM.
Potassium carbonate-mediated
efficient and convenient
synthesis
3-Methyl-1-phenylchromeno[4,3-c]pyrazol-4(1H)-ones.
Synthetic Communications
2014, 44: 1914-23. |
 |
Grover J, Kumar
V, Sobhia ME and Jachak SM.
Synthesis, biological evaluation
and docking analysis of
3-Methyl-1-phenylchromeno[4,3-c]pyrazol-4(1H)-ones
as potential cyclooxygenase
(COX)-2 inhibitors.
Bioorganic and Medicinal
Chemistry Letters 2014,
24:4638-42. |
 |
Bahl A, Jachak
SM, Palaniveloo K, Ramachandram
T, Vairappan CS and Chopra HK.
2-Acetoxyverecynarmin C, a new
briarane COX inhibitory
diterpenoid from Pennatula
aculeata. Natural Products
Communications 2014, 9: 1139-41. |
 |
Chandna N, Kapoor
JK, Grover J, Bairwa K, Goyal V
and Jachak SM.
Pyrazolylbenzyltriazoles as
cyclooxygenase inhibitors:
synthesis and biological
evaluation as dual
anti-inflammatory and
antimicrobial agents. New
Journal of Chemistry
2014, 38: 3662-72. |
 |
Mishra S, Aeri V,
Gaur PK
and
Jachak SM. Phytochemical,
therapeutic and
Ethnopharmacological Overview of
a Traditionally Important Herb:
Boerhavia diffusa Linn.
Biomedical Research
International
2014,
2014:
Article ID 808302: 19 pages (http://dx.doi.org/10.1155/2014/808302). |
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Kaur A, Kaur PK,
Singh S
and
Singh IP.
Antileishmanial
compounds from Moringa
oleifera Lam.
Zeitschrift fuer Naturforschung
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2014, 69c:
110-16. |
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Aqil F, Vadhanam
MV, Jeyabalan J, Cai J, Singh IP
and
Gupta RC.
Detection of
anthocyanins/anthocyanidins in
animal tissues. J. Agric.
Food Chem. 2014,
62: 3912-18. |
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Mahajan S,
Khullar S, Mandal S and Singh
IP. A one-pot, three-component
reaction for the synthesis of
novel 7-arylbenzo[c]acridine-5,6-diones
ChemComm.,
2014 , 50: 10078-81. |
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Aqil F, Munagala R, Jeyabalan J,
Joshi T, Singh IP
and
Gupta RC. The Indian Blackberry
(Jamun), Antioxidant Capacity,
and Cancer Protection
In: Victor R Preedy (Ed)
Cancer: Oxidative Stress and
Dietary Antioxidants 2014.
Elsevier Academic Press USA.
100-114. |
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Singh IP and Sidana J. Chemistry
of the genus Eucalyptus.
In Bhojvaid et al (Eds)
Eucalypts in India,
ENVIS centre on Forestry, FRI,
Dehradun, India. 2014,
429-69. |
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Dhillon RS, Singh IP and Baskar
C. 2014, STEREOCHEMISTRY,
ISBN: 9788184872415,
Narosa Publications, New Delhi. |
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Kumar V and Sobhia ME. Insights
into the bonding pattern for
characterizing the open and
closed state of the
substrate-binding loop in
Mycobacterium tuberculosis InhA.
Future Med Chem.
2014, 6: 605-16. |
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Grewal BK,
Krishnan RV and Sobhia ME.
Structural basis
of conformational variance in
phosphorylated and non-phosphorylated
states of PKCβII.
Proteins 2014,
7: 1332-47. |
 |
Anand B and
Sobhia ME. Exploring a model of
human chemokine receptor CCR2 in
presence of TAK779: A membrane
based molecular dynamics study.
Journal of Molecular
Structure 2014, 1063:
131-38. |
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Grewal, BK and
Sobhia ME. Scaffold Hopping for
Identification of Novel PKCβII
Inhibitors Based on Ligand and
Structural Approaches, Virtual
Screening and Molecular Dynamics
Study.
Combinatorial
Chemistry & High Throughput
Screening
2014, 17: 2-11. |
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Khan S and Jena
GB. Sodium butyrate, a HDAC
inhibitor ameliorates eNOS, iNOS
and TGF-beta1-induced
fibrogenesis, apoptosis and DNA
damage in the kidney of juvenile
diabetic rats. Food and
Chemical Toxicology
2014, 73: 127-139. |
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Parmar AR,
Trivedi PP and Jena GB. Dextran
sulfate sodium-induced
ulcerative colitis leads to
testicular toxicity in mice:
Role of inflammation, oxidative
stress and DNA damage.
Reproductive Toxicology
2014, 49: 171-184. |
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Yadav L, Khan S
and Jena GB. Influence of
3-Aminobenzamide, a PARP
inhibitor in the genotoxicity
evaluation of selected
candidates. Mutation
Research 2014, 770: 6-15. |
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Shekh K, Khan S,
Jena GB, Kansara B and Kushwaha
S. 3-aminobenzamide, a PARP
inhibitor enhances the
sensitivity of peripheral blood
micronucleus and comet assays in
mice. Toxicology
Mechanisms and Methods
2014, 24(5): 332-341. |
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Maremanda KP,
Khan S, Jena GB. Zinc
protects
cyclophosphamide-inducedtesticular
damage in rat: involvement of
metallothionein, tesmin and
Nrf2. Biochemical and
Biophysical Research
Communications 2014,
445(3): 591-6. |
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Khan S and Jena
GB. Protective role of sodium
butyrate, a HDAC inhibitor on
beta-cell proliferation,
function and glucose homeostasis
through modulation of p38/ERK
MAPK and apoptotic pathways:
Study in juvenile diabetic rat.
Chemico Biological
Interaction 2014, 213:
1-12. |
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Khan S and Jena
GB. Sodium valproate, a histone
deacetylase inhibitor
ameliorates cyclophosphamide-induced
genotoxicity and cytotoxicity in
the colon of mice. Journal
Basic Clinical Physiology and
Pharmacology 2014, 27:
1-11. |
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Jena GB and
Trivedi PP. A review of the use
of melatonin in ulcerative
colitis: Experimental evidence
and new approaches .
Inflammatory Bowel Disease
2014, 20(3): 553-63. |
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Angrish, Anil Kumar and Bansal,
S. K. Private Sector Banking in
India: A Perspective.
Latest Trends in Management,
Commerce & Economics: A
Collection of Research Papers
ISBN: 978-81-928584-1-8. 2014:
101-06. |
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Bajaj P, Tripathy RK, Aggarwal
G, and Pande AH. Paraoxonase 1
as a pharmacologic agent:
limitations and perspectives.
The Scientific World
Journal.1 2014, 2014. |
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Bajaj P, Tripathy RK, Aggarwal
G, Pande AH. Interplay between
amino acid residues at positions
192 and 115 in modulating
hydrolytic activities of human
paraoxonase 1. Biochimie
2014, 105: 202-10. |
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Bajaj P, and Pande AH.
Stabilization studies on
bacterially produced human
paraoxonase1 for improving its
shelf life. Appl. Biochem.
Biotechnol. 2014,
172: 3798-809. |
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Nankar SA, Pande AH. Properties
of apolipoprotein E derived
peptide modulate their
lipid-binding capacity and
influence their
anti-inflammatory function.
Biochim Biophys Acta. 2014,
1841: 620-29. |
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Nankar SA, Prajapati JS, Pande
AH. Apolipoprotein E derived
peptides inhibit the
pro-inflammatory effect of
lysophosphatidylcholine.
Protein Pept. Lett.
2014, 21: 101-07. |
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Guchhait S,
Priyadarshani G and Hura N.
α,β-Epoxy Esters in Multiple
C–O/C–N Bond-Breaking/Formation
with 2-Aminopyridines; Synthesis
of Biologically Relevant
(Z)-2-Methylene-imidazo[1,2-a]pyridin-3-ones.
Synlett
2014, 25: 1692-96. |
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Sanghai N, Jain
V, Preet R, Kandekar S, Das S,
Trivedi N, Mohaputra P,
Priyadarshani G, Kashyap M, Das
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Sheokand N,
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Harde H, Agrawal
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Journal of
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Sonawane R, Harde
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Nanoparticles Loaded Topical Gel
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Expert Opinion on Drug
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Kulthe S, Inamdar
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Agrawal M, Agrawal SK, Jain S
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Nanocarriers for Controlled and
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Journal of
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Jain S,
Jain R, Das M, Agrawal AK,
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Combinatorial Bio-Conjugation of
Gemcitabine and Curcumin Enables
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and Reduced Toxicity. RSC
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Swarnakar NK,
Thanki K and Jain S. Enhanced antitumor efficacy and
counterfeited cardiotoxicity of
combinatorial oral therapy using
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Q10-liquid crystalline
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and Medicine
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Swarnakar NK,
Thanki K and Jain S. Lyotropic
liquid crystalline nanoparticles
of CoQ10: Implication of
lipase-digestibility on oral
bioavailability, in vivo
antioxidant activity and
in-vitro in-vivo relationships.
Molecular Pharmaceutics
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Das M, Jain R,
Agrawal AK, Thanki K and Jain S.
Macromolecular bipill of
gemcitabine and methotrexate
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drug therapy with higher
benefit-to-risk ratio.
Bioconjugate Chemistry
2014, 25: 501-09. |
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Jain AK, Thanki
K and Jain S. Novel self-nanoemulsifying
formulation of quercetin:
Implications of pro-oxidant
activity on the anticancer
efficacy.
Nanomedicine: Nanotechnology, Biology
and Medicine
2014, 10: 959-69. |
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Swarnakar NK,
Thanki K and Jain S.
Bicontinuous cubic liquid
crystalline nanoparticles for
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therapeutic efficacy and
cardiotoxicity.
Pharmaceutical Research
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Jain AK, Thanki
K and Jain S. Solidified self-nanoemulsifying
formulation for oral delivery of
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antitumor efficacy and
hepatotoxicity.
Pharmaceutical Research
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Jain AK, Thanki K
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self-nanoemulsifying formulation
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Jain S, Harde H,
Indulkar A and Agrawal AK. Improved
stability and immunological
potential of tetanus toxoid
containing surface engineered
bilosomes following oral
administration.
Nanomedicine: Nanotechnology, Biology
and Medicine
2014, 10: 431-40. |
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Jain S, Indulkar
A, Harde H and Agrawal AK. Oral
mucosal immunization using
glucomannosylated bilosomes.
Journal of Biomedical
Nanotechnology 2014, 10:
932-47. |
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Agrawal AK, Harde
H, Thanki K and Jain S.
Improved stability and
antidiabetic potential of
insulin containing folic acid
functionalized polymer
stabilized multilayered
liposomes following oral
administration.
Biomacromolecules 2014,
15: 350-60. |
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Dinesh N,
Pallerla DS, Kaur PK, Babu NK
and Singh S. Exploring
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3-hydroxy-3-methylglutaryl
coenzyme A reductase (HMGR) as a
potential drug target by
biochemical, biophysical and
inhibition studies.
Microbial Pathogenesis
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Kaur A, Kaur PK,
Singh S and Singh IP.
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Zeitschrift für Naturforschung.
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Singh S, Dinesh
N, Kaur PK and Shamiulla B.
Ketanserin, an antidepressant
exerts its antileishmanial
action via inhibition of
3-hydroxy-3-methylglutaryl
coenzyme A reductase (HMGR)
enzyme of Leishmania donovani.
Parasitology Research 2014, 113(6):
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Singh S, Raju K,
Jatekar D, Dinesh N, Paul MS and
Sobhia ME. Leishmania
donovani eukaryotic
initiation factor 5A: Molecular
characterization, localization
and homology modelling studies.
Microbial Pathogenesis
2014, 73: 37-46. |
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Dinesh N, Kaur PK,
Swamy KK and Singh S. Mianserin,
an antidepressant kills
Leishmania donovani by
depleting ergosterol levels.
Experimental Parasitology
2014, 144: 84-90. |
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Kaur PK, Supin JK,
Rashmi S and Singh S. Chemical
and thermal induced unfolding of
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A single tryptophan protein.
Applied Biochemistry and
Biotechnology2014, 173:
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Bhagat S, Shah P,
Garg SK, Mishra S,
Kaur PK, Singh
S and Chakraborti AK. α-Aminophosphonates
as novel anti-leishmanial
chemotypes: synthesis,biological
evaluation, and CoMFA studies.
Medicinal Chemistry
Communications 2014,
5:
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Tumbi M,
Nandedkar P, Naeem Shaikh, Kesharwani
S and Sangamwar A. Molecular
dynamics simulation studies for
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reactive metabolites of
anticancer compounds. J
Molecular Recognition
2014, 27: 138-50. |
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Khandelwal K,
Gangwal R, Singh U, Prajapati R,
Damre M and Sangamwar A.
Computational insights into the
active site of human breast
cancer resistance protein (BCRP/ABCG2):
A similarity search approach.
Med Chem Res. 2014,
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Kumar V,
Rachamalla M, Nandekar P,
Khatik G, Sangamwar A,
Tikoo K
and
Nair V. Design and synthesis of
optically pure
3-aryl-6-methyl-2-thiooxotetrahydropyrimidin-4(1H)-ones
as anti-prostate cancer agents,
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Rathod V, Jain S,
Nandekar P and Sangamwar A. Human
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Uppalapati D, Das
N, Gangwal R, Damre M, Sangamwar
A and Sharma S. Neuroprotective
Potential of Peroxisome
Proliferator Activated
receptor-α (PPAR-α) agonist in
cognitive impairment in
Parkinson’s disease: Behavioral,
biochemical and PBPK profile.
PPAR Research 2014,
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Damre M, Gangwal
R, Dhoke G, Lalit M, Sharma D,
Khandelwal K and Sangamwar A. 3D
QSAR and molecular docking
studies of aminopyrimidine
derivatives as PknB inhibitors.
J of Taiwan Institute of
Chemical Engineers 2014,
45: 354-364. |
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Dara A and
Sangamwar A. Identifying the
Patent Trend, Licensing Pattern
and Geographical Landscape
Analysis of the Council for
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2011.
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1. Yadav
I, Nandekar P, Shrivastava S,
Sangamwar A, Chaudhary A
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knoevenagelcurcumin derivatives
with potent anti-EGFR activity.
Gene
2014,
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1. Kalariya
P, Raju B, Borkar R, Namdev D,
Gananadhamu
S, Nandekar P, Sangamwar A and
Srinivas R. Characterization of
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ketorolac tromethamine using LC/ESI/Q/TOF/MS/MS
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J of Mass Spectrometry.
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1. Pragyan
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Predicting drug metabolism by
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insights from MetaSite,
molecular docking and quantum
chemical calculations.
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Prajapati R and Sangamwar A.
Translocation mechanism of
P-glycoprotein and
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at drug binding site: Insights
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Dynamics.
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Dara A and Sangamwar A. Clearing
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Nandekar P
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P-glycoprotein: a connexion for
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Mol. Divers 2014,
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Kesharwani S,
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Gangwal
R, Damre M, Das N,
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Bansal D, Gudala
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diabetes mellitus in a tertiary
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Ghai B, Bansal D,
Kay JP, Vadaje KS and Wig J. Transforaminal versus
parasagittal interlaminar
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low back pain with radicular
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Kanukula R,
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Kumar S, Bansal
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clinical outcomes and
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inpatients with severe
preeclampsia and eclampsia: an
Indian experience. Indian
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Ghai B, Jain K,
Bansal D and Wig J. End-tidal
concentrations of sevoflurane
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Savla JR, Ghai B,
Bansal D and Wig J. Effect of
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oral midazolam premedication on
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laryngeal mask airway placement
in children: a randomized,
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Kapil G, Bansal D
and Ghai B. Missing values in
patient reported outcomes:
assessment of disability in
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Pain Physician 2014,
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Ghai B, Bansal D,
Hota D and Shah CS. Off-label,
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Bansal D, Gudala
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RV and Bhansali A.
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Mellitus Patients.
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Choubey AK,
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Activity. Bioorganic
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Jain SK, Gill
MS, Pawar HS and Suresh S. Novel
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Enhanced Curcumin Bioavailbility
and Efficacy in Streptococcal
Cel Wall-induced Arthritis.
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Singh C,
Joydev L, Bhatt TD, Gill MS and
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biochemical and
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Laha JK, Dayal N, Jain R and
Patel K. Palladium-Catalyzed
Regiocontrolled Domino Synthesis
of N-Sulfonyl
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Dihydrodibenzo[c,e]azepines:
Control over the Formation of
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Laha JK, Jethava KP, Dayal
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Intramolecular Oxidative
Coupling Involving Double
C(sp2)–H Bonds for the Synthesis
of Annulated Biaryl Sultams.
J. Org. Chem.
2014, 79: 8010–19. |
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Laha JK,
Tummalapalli KSS and Gupta
A. Transition-Metal-Free Tandem
Oxidative Removal of Benzylic Methylene
Group by C–C and C–N Bond
Cleavage Followed by
Intramolecular New Aryl C–N Bond
Formation under Radical
Conditions. Org. Lett., 2014, 16: 4392–95. |
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Laha JK, Dayal N,
Singh S and Bhimpuria R. Dual
Catalysis in Domino N-Benzylation/Intramolecular
C–H Arylation: Regio- and
Chemoselective Synthesis of
Annelated Nitrogen Heterocycles.
Eur. J. Org. Chem.
2014, 5469-75. |
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Laha JK,
Tummalapalli KSS and Gupta A.
Mechanistic Insights into the
Palladium-Catalyzed Domino
Synthesis of
10,11-Dihydro-5H-dibenzo[b,e][1,4]diazepines
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